2883653-86-7
Chemical Structure
Helianorphin-19
- CAS No.: 2883653-86-7
- Formula:C81H132N26O16S2
- Molecular Weight:1790.21
InChIKey: WEJHFJXWIBZZTQ-AHUOXLFJSA-N
SMILES: O=C([C@@H](NC1=O)CSSC[C@H](NC2=O)C(N[C@H](C(N[C@H](C(N3[C@H](C(N[C@H](C(N[C@H](C(N[C@H]1CCCCN)=O)CC(C)C)=O)CCCCN)=O)CCC3)=O)CCCNC(N)=N)=O)[C@H](CC)C)=O)N[C@H](C(NCC(NCC(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H]2CCCNC(N)=N)=O)CCCNC(N)=N)=O)CC(C)C)=O)CC4=CC=CC=C4)=O)=O)=O)CC5=CC=C(O)C=C5
Biological Activity: Helianorphin-19 is a potent and selective κ-opioid receptor (KOR) activator with a Ki of 21 nM and an EC50 of 45 nM. Helianorphin-19 exhibits strong KOR-specific peripheral analgesic activity in a mouse model of chronic visceral pain[1].
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Helianorphin-19 | Helianorphin-19 is a potent and selective κ-opioid receptor (KOR) activator with a Ki of 21 nM and an EC50 of 45 nM. Helianorphin-19 exhibits strong KOR-specific peripheral analgesic activity in a mouse model of chronic visceral pain. | |||||||||||||||||||||
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