3082554-75-1
3082554-75-1
Chemical Structure
BI-9508
- CAS No.: 3082554-75-1
- Formula:C28H29F2N5O3
- Molecular Weight:521.56
InChIKey: BZJPCUQQPJJBTP-FGZHOGPDSA-N
SMILES: CC(C)OC1=CC=C(C2=C3C(N(C)N=C3)=C(N(CCOC(F)F)C([C@H]4[C@H](C5=CC=NC=N5)C4)=O)C=C2)C=C1
Biological Activity: BI-9508 is a blood-brain barrier-penetrant GPR88 agonist. BI-9508 acts through activation of the Gi1 signaling pathway; it exists as atropisomers, with the more active isomer showing stronger agonist potency and lower P-glycoprotein efflux. BI-9508 can be used in GPR88-related central nervous system research[1].
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BI-9508 | BI-9508 is a blood-brain barrier-penetrant GPR88 agonist. BI-9508 acts through activation of the Gi1 signaling pathway; it exists as atropisomers, with the more active isomer showing stronger agonist potency and lower P-glycoprotein efflux. BI-9508 can be used in GPR88-related central nervous system research. | |||||||||||||||||||||
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