3136748-24-5
3136748-24-5
Chemical Structure
TGF-8027
- CAS No.: 3136748-24-5
- Formula:C19H22N2O3
- Molecular Weight:326.39
InChIKey: YGVDYCKUVCKBFS-UHFFFAOYSA-N
SMILES: COC1=C(CCNC(C)C2=CC=CC=C2O)C=C(OC)C(C#N)=C1
Biological Activity: TGF-8027 is a selective 5-HT2A receptor agonist with a Ki of 7.4 nM and an EC50 of 3.3 nM at the human receptor. TGF-8027 activates the 5-HT2A receptor-mediated Gq protein signaling pathway. TGF-8027 induces dose-dependent head-twitch responses in mice[1].
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TGF-8027 | TGF-8027 is a selective 5-HT2A receptor agonist with a Ki of 7.4 nM and an EC50 of 3.3 nM at the human receptor. TGF-8027 activates the 5-HT2A receptor-mediated Gq protein signaling pathway. TGF-8027 induces dose-dependent head-twitch responses in mice. | |||||||||||||||||||||
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