330834-54-3
Chemical Structure
AGX51
- CAS No.: 330834-54-3
- Formula:C27H29NO4
- Molecular Weight:431.52
IUPAC Name: N-(3-(benzo[d][1,3]dioxol-5-yl)-3-(2-methoxyphenyl)propyl)-N-benzylpropionamide
InChIKey: SRADCMOCDMFMPS-UHFFFAOYSA-N
SMILES: CCC(N(CCC(C1=CC=C(OCO2)C2=C1)C3=CC=CC=C3OC)CC4=CC=CC=C4)=O
Biological Activity: AGX51 is the first-in-class pan-Id (inhibitors of DNA-binding/differentiation proteins) antagonist and degrader. AGX51 inhibits Id1-E47 interaction, leading to ubiquitin-mediated degradation of Ids, cell growth arrest, and viability reduction. AGX51 can inhibit TNBC and has an IC50 of about 25 nM. AGX51 can be used in cancer research.
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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AGX51 | 99.33% | AGX51 is the first-in-class pan-Id (inhibitors of DNA-binding/differentiation proteins) antagonist and degrader. AGX51 inhibits Id1-E47 interaction, leading to ubiquitin-mediated degradation of Ids, cell growth arrest, and viability reduction. AGX51 can inhibit TNBC and has an IC50 of about 25 nM. AGX51 can be used in cancer research. | ||||||||||||||||||||
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Keywords
