56173-05-8
56173-05-8
Chemical Structure
PCAF-IN-2
- CAS No.: 56173-05-8
- Formula:C10H7F3N6
- Molecular Weight:268.20
IUPAC Name: 6-hydrazinyl-3-(trifluoromethyl)-[1,2,4]triazolo[3,4-a]phthalazine
InChIKey: VXUZXROYRSNHSD-UHFFFAOYSA-N
SMILES: FC(C1=NN=C2N1N=C(NN)C3=C2C=CC=C3)(F)F
Biological Activity: PCAF-IN-2 (compound 17) is a potent PCAF inhibitor with an IC50 value of 5.31 µM. PCAF-IN-2 shows anti-tumour activity. CAF-IN-2 induces apoptosis and arrest the cell cycle at the G2/M phase[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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PCAF-IN-2 | 98.0% | PCAF-IN-2 (compound 17) is a potent PCAF inhibitor with an IC50 value of 5.31 µM. PCAF-IN-2 shows anti-tumour activity. CAF-IN-2 induces apoptosis and arrest the cell cycle at the G2/M phase. | ||||||||||||||||||||
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Structural Analogs
-
Similarity Score 0.60
HY-179573UCM-A86 -
Similarity Score 0.58
HY-103505RCL 218872 (Standard) -
Similarity Score 0.58
HY-147894PCAF-IN-1 -
Similarity Score 0.55
HY-1345616-Amino-8-trifluoromethylphenanthridine -
Similarity Score 0.55
HY-155078BRD4 Inhibitor-27 -
Similarity Score 0.53
HY-12593GS967 -
Similarity Score 0.52
HY-124859CeMMEC2 -
Similarity Score 0.52
HY-119057DSM74 -
Similarity Score 0.51
HY-B1001ATodralazine hydrochloride -
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