700878-19-9
700878-19-9
Chemical Structure
NMDA-IN-1
- CAS No.: 700878-19-9
- Formula:C20H23ClFN3O
- Molecular Weight:375.87
IUPAC Name: 2-((4-(2-fluorobenzyl)piperidin-1-yl)methyl)-1H-benzo[d]imidazol-6-ol hydrochloride
InChIKey: IJHXPTYEGXYLBZ-UHFFFAOYSA-N
SMILES: OC1=CC=C2N=C(CN3CCC(CC4=CC=CC=C4F)CC3)NC2=C1.[H]Cl
Biological Activity: NMDA-IN-1 is a potent and NR2B-selective NMDA antagonist with Ki of 0.85 nM; NR2B Ca2+ influx IC50 is 9.7 nM; no activities on NR2A, NR2C, NR2D, hERG-channel and α1-adrenergic receptor.
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
|
|
NMDA-IN-1 | 98.98% | NMDA-IN-1 is a potent and NR2B-selective NMDA antagonist with Ki of 0.85 nM; NR2B Ca2+ influx IC50 is 9.7 nM; no activities on NR2A, NR2C, NR2D, hERG-channel and α1-adrenergic receptor. | ||||||||||||||||||||
|
loading...
/
|
|||||||||||||||||||||||
Keywords
