1. Membrane Transporter/Ion Channel
    Neuronal Signaling
  2. iGluR
  3. NMDA-IN-1

NMDA-IN-1 

Cat. No.: HY-12962 Purity: >98.0%
Handling Instructions

NMDA-IN-1 is a potent and NR2B-selective NMDA antagonist with Ki of 0.85 nM; NR2B Ca2+ influx IC50 is 9.7 nM; no activities on NR2A, NR2C, NR2D, hERG-channel and α1-adrenergic receptor.

For research use only. We do not sell to patients.

NMDA-IN-1 Chemical Structure

NMDA-IN-1 Chemical Structure

CAS No. : 700878-19-9

Size Price Stock Quantity
10 mM * 1 mL in DMSO USD 308 In-stock
Estimated Time of Arrival: December 31
5 mg USD 280 In-stock
Estimated Time of Arrival: December 31
10 mg USD 480 In-stock
Estimated Time of Arrival: December 31
50 mg   Get quote  
100 mg   Get quote  

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Description

NMDA-IN-1 is a potent and NR2B-selective NMDA antagonist with Ki of 0.85 nM; NR2B Ca2+ influx IC50 is 9.7 nM; no activities on NR2A, NR2C, NR2D, hERG-channel and α1-adrenergic receptor.

Molecular Weight

375.87

Formula

C₂₀H₂₃ClFN₃O

CAS No.

700878-19-9

SMILES

OC1=CC=C2N=C(CN3CCC(CC4=CC=CC=C4F)CC3)NC2=C1.[H]Cl

Shipping

Room temperature in continental US; may vary elsewhere.

Storage
Powder -20°C 3 years
4°C 2 years
In solvent -80°C 6 months
-20°C 1 month
References
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Keywords:

NMDA-IN-1iGluRIonotropic glutamate receptorsInhibitorinhibitorinhibit

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NMDA-IN-1
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