844639-57-2
Chemical Structure
CAY10471 Racemate
Synonym(s): TM30089 Racemate
- CAS No.: 844639-57-2
- Formula:C21H21FN2O4S
- Molecular Weight:416.47
IUPAC Name: 2-(3-((4-fluoro-N-methylphenyl)sulfonamido)-1,2,3,4-tetrahydro-9H-carbazol-9-yl)acetic acid
InChIKey: CANCTKXGRVNXFP-UHFFFAOYSA-N
SMILES: O=C(O)CN1C2=C(C3=C1C=CC=C3)CC(N(S(=O)(C4=CC=C(F)C=C4)=O)C)CC2
Biological Activity: CAY10471 Racemate (TM30089 Racemate) is a potent and highly selective prostaglandin D2 receptor CRTH2 antagonist, with a Ki of 0.6 nM for hCRTH2, selective over human thromboxane A2 receptor TP (Ki, >10000 nM) or PGD2 receptor DP (Ki, 1200 nM). CAY10471 Racemate also has effect on mouse and rat orthologs of CRTH2[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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CAY10471 Racemate | 99.00% | CAY10471 Racemate (TM30089 Racemate) is a potent and highly selective prostaglandin D2 receptor CRTH2 antagonist, with a Ki of 0.6 nM for hCRTH2, selective over human thromboxane A2 receptor TP (Ki, >10000 nM) or PGD2 receptor DP (Ki, 1200 nM). CAY10471 Racemate also has effect on mouse and rat orthologs of CRTH2. | ||||||||||||||||||||
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