86329-06-8
Chemical Structure
CP59430
- CAS No.: 86329-06-8
- Formula:C21H22N8O3
- Molecular Weight:434.45
IUPAC Name: (4-(4-amino-6,7-dimethoxyquinazolin-2-yl)piperazin-1-yl)(4-azidophenyl)methanone
InChIKey: XHCZPSMUDVXSPQ-UHFFFAOYSA-N
SMILES: COC1=CC2=NC(N3CCN(C(C4=CC=C(N=[N+]=[N-])C=C4)=O)CC3)=NC(N)=C2C=C1OC
Biological Activity: CP59430 is an azide analog of the α-adrenaline receptor antagonist Prazosin (HY-B0193). P59430 behaves as a competitive antagonist of α1-adrenaline receptor before photolysis. After photolysis, it specifically and irreversibly labels α1-adrenaline receptor and exhibits non-competitive antagonist activity. CP59430 can be used for the study of receptor molecular characterization[1].
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CP59430 | CP59430 is an azide analog of the α-adrenaline receptor antagonist Prazosin (HY-B0193). P59430 behaves as a competitive antagonist of α1-adrenaline receptor before photolysis. After photolysis, it specifically and irreversibly labels α1-adrenaline receptor and exhibits non-competitive antagonist activity. CP59430 can be used for the study of receptor molecular characterization. | |||||||||||||||||||||
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Keywords
