91406-11-0
91406-11-0
Chemical Structure
Esuprone
- CAS No.: 91406-11-0
- Formula:C13H14O5S
- Molecular Weight:282.31
IUPAC Name: 3,4-dimethyl-2-oxo-2H-chromen-7-yl ethanesulfonate
InChIKey: CHDGAVDQRSPBTA-UHFFFAOYSA-N
SMILES: CC(C1=CC=C(OS(CC)(=O)=O)C=C1O2)=C(C)C2=O
Biological Activity: Esuprone is a brain-penetrant, orally active and selective MAO A inhibitor with an IC50 of 7.3 nM. Esuprone can be used for neurological research[1][2].
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Esuprone | 99.67% | Esuprone is a brain-penetrant, orally active and selective MAO A inhibitor with an IC50 of 7.3 nM. Esuprone can be used for neurological research. | ||||||||||||||||||||
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References
- [1]. Löscher W, et al. Inhibition of monoamine oxidase type A, but not type B, is an effective means of inducing anticonvulsant activity in the kindling model of epilepsy. J Pharmacol Exp Ther. 1999 Mar;288(3):984-92. [Content Brief]
- [2]. Bergström M, et al. MAO-A inhibition in brain after dosing with esuprone, moclobemide and placebo in healthy volunteers: in vivo studies with positron emission tomography. Eur J Clin Pharmacol. 1997;52(2):121-8. [Content Brief]
Keywords
