936501-01-8
936501-01-8
Chemical Structure
Elinogrel potassium
Synonym(s): PRT060128 potassium
- CAS No.: 936501-01-8
- Formula:C20H15ClFKN5O5S2
- Molecular Weight:563.04
IUPAC Name: 5-chloro-N-((4-(6-fluoro-7-(methylamino)-2,4-dioxo-1,2-dihydroquinazolin-3(4H)-yl)phenyl)carbamoyl)thiophene-2-sulfonamide, potassium salt
InChIKey: PUTUVTXPBZTQMO-UHFFFAOYSA-N
SMILES: O=S(C1=CC=C(Cl)S1)(NC(NC2=CC=C(N3C(NC4=C(C=C(F)C(NC)=C4)C3=O)=O)C=C2)=O)=O.[K]
Biological Activity: Elinogrel (PRT060128) potassium is a reversible, competitive and orally active P2Y12 antagonist. Elinogrel potassium inhibits thrombosis[1][2].
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Elinogrel potassium | Elinogrel (PRT060128) potassium is a reversible, competitive and orally active P2Y12 antagonist. Elinogrel potassium inhibits thrombosis. | |||||||||||||||||||||
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References
- [1]. Ueno M, et al. Elinogrel: pharmacological principles, preclinical and early phase clinical testing. Future Cardiol. 2010 Jul;6(4):445-53. [Content Brief]
- [2]. Haberstock-Debic H, et al. A clopidogrel-insensitive inducible pool of P2Y12 receptors contributes to thrombus formation: inhibition by elinogrel, a direct-acting, reversible P2Y12 antagonist. J Pharmacol Exp Ther. 2011 Oct;339(1):54-61. [Content Brief]
Keywords
