872002-72-7
872002-72-7
Chemical Structure
WAY-207024
- CAS. Nr.: 872002-72-7
- Formula:C30H32N6
- Molecular Weight:476.62
IUPAC Name: 6-((4-(2-(4-(tert-butyl)phenyl)-1H-benzo[d]imidazol-7-yl)piperazin-1-yl)methyl)quinoxaline
InChIKey: AVEVJMZJJJDOCI-UHFFFAOYSA-N
SMILES: CC(C1=CC=C(C2=NC3=CC=CC(N4CCN(CC5=CC=C6N=CC=NC6=C5)CC4)=C3N2)C=C1)(C)C
Biological Activity: WAY-207024 is an orally active gonadotropin releasing hormone receptor (GnRH-R) antagonist (human GnRH: IC50 of 12 nM, rat GnRH: IC50 of 71 nM). WAY-207024 inhibits rat LH release with an IC50 of 350 nM. WAY-207024 lowers rat plasma leuteinizing hormone (LH) levels after oral administration[1].
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WAY-207024 | WAY-207024 is an orally active gonadotropin releasing hormone receptor (GnRH-R) antagonist (human GnRH: IC50 of 12 nM, rat GnRH: IC50 of 71 nM). WAY-207024 inhibits rat LH release with an IC50 of 350 nM. WAY-207024 lowers rat plasma leuteinizing hormone (LH) levels after oral administration. | |||||||||||||||||||||
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