PSI-112
PSI-112 is a YO-class μPlm inhibitor, with IC50 values of 0.38 μM, 1.48 μM and 0.37 μM against the wild-type, F587A mutant and K607A mutant, respectively. PSI-112 shows low affinity for uPA. PSI-112 can be used in cancer research.
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- No. CAS: 1854997-77-5
- Fòrmula: C35H48N4O3
- Peso molecular:572.78
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Actividad biológica
Descripciòn
IC50 & Target
[1]|
μPlm 0.38 μM (IC50) |
In Vitro
PSI-112 inhibits wild-type μPlm with an IC50 of 0.38 μM, and its affinity for uPA (IC50 >25 μM) is lower than that for μPlm[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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No. CAS 1854997-77-5
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Peso molecular 572.78
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Fòrmula C35H48N4O3
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SMILES
O=C([C@@H]1CC[C@H](CC1)CN)N[C@H](C(NCCCCCCCC)=O)CC(C=C2)=CC=C2OCC3=NC4=C(C=CC=C4)C=C3
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
PSI-112 Related Classifications
HY-182565 Related Classifications
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