PF-184563
Janthitrem F is a metabolite isolated from tremorigen-producing Penicillium and a potential causative agent of ryegrass spurt disease.
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- CAS 番号: 748806-39-5
- 分子式: C21H23ClN6
- 分子量:394.90
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保管条件:
Please store the product under the recommended conditions in the Certificate of Analysis.
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生物活性
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化学情報
- 純度とドキュメンテーション
- 参考文献
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Help & FAQs
生物活性
製品説明
IC50 & Target
Penicillium sp.[1]
Cellular Effect
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| CHO | IC50 |
6.7 nM
Compound: 13d, PF-184563
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Antagonist activity at human V1A receptor expressed in CHO cells assessed as inhibition of AVP-induced intracellular calcium release after 30 seconds by FLIPR assay
Antagonist activity at human V1A receptor expressed in CHO cells assessed as inhibition of AVP-induced intracellular calcium release after 30 seconds by FLIPR assay
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[PMID: 21885275] |
| HEK293 | IC50 |
17900 nM
Compound: 13d, PF-184563
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Displacement of [3H]dofetilide from human ERG transfected in HEK293 cells by fluorescence polarization binding assay
Displacement of [3H]dofetilide from human ERG transfected in HEK293 cells by fluorescence polarization binding assay
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[PMID: 21885275] |
化学情報
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CAS 番号 748806-39-5
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分子量 394.90
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分子式 C21H23ClN6
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SMILES
CN1CC2=CC(Cl)=CC=C2N3C(C4CCN(CC4)C5=NC=CC=C5)=NN=C3C1
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
Please store the product under the recommended conditions in the Certificate of Analysis.
純度とドキュメンテーション
参考文献
Calculators
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)
PF-184563 関連分類
HY-121163 関連分類
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