PI3Kδ-IN-9
PI3Kδ-IN-9 is a selective PI3Kδ inhibitor with an IC50 value of 3.8 nM.
For research use only. We do not sell to patients.
- CAS No.: 2135922-40-4
- Formula: C24H26FN9O
- Molecular Weight:475.52
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| HeLa | IC50 |
5.4 μM
Compound: 4d; L-006021422
|
Inhibition of [3H]adenosine uptake in human HeLa cells preincubated for 30 mins followed by incubation with [3H]adenosine for 60 mins by TopCount plate reader analysis
Inhibition of [3H]adenosine uptake in human HeLa cells preincubated for 30 mins followed by incubation with [3H]adenosine for 60 mins by TopCount plate reader analysis
|
[PMID: 33335668] |
Chemical Information
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CAS No. 2135922-40-4
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Molecular Weight 475.52
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Formula C24H26FN9O
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SMILES
O=C1[C@@](C)(NCC(C)(F)C)C2=CC(C3=C4N=C(C5=CN=C(C)N=C5)N(CC)C4=NC=N3)=CN=C2N1
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)