1. Antibody-drug Conjugate/ADC Related
    PROTAC
  2. PROTAC-linker Conjugate for PAC
  3. PROTAC BRD4 degrader for PAC-1

PROTAC BRD4 degrader for PAC-1 

Cat. No.: HY-129938
Handling Instructions

PROTAC BRD4 degrader for PAC-1 (compound 5), a PROTAC-linker Conjugate for PAC, comprises the chimeric BET degrader GNE-987 and disulfide-containing linker.

For research use only. We do not sell to patients.

PROTAC BRD4 degrader for PAC-1 Chemical Structure

PROTAC BRD4 degrader for PAC-1 Chemical Structure

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Description

PROTAC BRD4 degrader for PAC-1 (compound 5), a PROTAC-linker Conjugate for PAC, comprises the chimeric BET degrader GNE-987 and disulfide-containing linker[1].

Molecular Weight

1306.58

Formula

C₆₂H₇₇F₂N₉O₁₂S₄

SMILES

O=C(C1=C(CS(=O)(C)=O)C=C(C(N(C2=NC=C(F)C=C2F)C3)=C1)C4=CN(C)C(C5=C4C3=CN5)=O)NCCCCCCCCCCC(N[[email protected]@H](C(C)(C)C)C(N6[[email protected]](C(NCC7=CC=C(C8=C(C)N=CS8)C=C7)=O)C[[email protected]@H](OC(OCC(C)(C)SS(C)(=O)=O)=O)C6)=O)=O

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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This equation is commonly abbreviated as: C1V1 = C2V2

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Keywords:

PROTAC BRD4 degrader for PAC-1PROTAC-linker Conjugate for PACPROTAC-linker for PROTAC-antibody ConjugateBRD4antibody-drugconjugatechimericproteindegraderdrugdeliveryInhibitorinhibitorinhibit

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Product name:
PROTAC BRD4 degrader for PAC-1
Cat. No.:
HY-129938
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