121 Results for "

ACAT

" in MedChemExpress (MCE) Product Catalog:
Products (121)

121 Results for "ACAT" in MCE Product Catalog:

  • Isoforms Recommended:
Cat. No.: HY-N10224
CAS No.: 156967-65-6
Terpendole C, produced by Albophoma yamanashiensis, shows potent inhibitory activity against acyl-CoA: cholesterol acyltransferase (ACAT) .
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Cat. No.: HY-N8331
CAS No.: 167612-17-1
Terpendole I is a fungal indole diterpenoid and an ACAT inhibitor (IC50 = 145 µM). Terpendole I can be used in studies related to lipid metabolism .
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Cat. No.: HY-RS00137
Research Areas:  

Others

Acat1 Mouse Pre-designed siRNA Set A contains three designed siRNAs for Acat1 gene (Mouse), as well as a negative control, a positive control, and a FAM-labeled negative control.

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Cat. No.: HY-124064
CAS No.: 128831-46-9
Target:  

Acyltransferase

Research Areas:  

Metabolic Disease

TMP-153 is an orally active inhibitor of ACAT with an IC50 value of approximately 5-10 nM against hepatic and intestinal ACAT in varicose animals. TMP-153 exhibits cholesterol-lowering effects and can be utilized in the research of atherosclerosis .
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Cat. No.: HY-129344
CAS No.: 96224-26-9
Target:  

Acyltransferase

Research Areas:  

Metabolic Disease

CL 277082 is a potent and selective acyl CoA:cholesterol acyltransferase (ACAT) inhibitor in microsomes. CL 277082 inhibits ACAT with IC50 values of 0.14 μM for intestinal mucosal microsomes, 0.74 μM for liver, and 1.18 μM for rat adrenal. CL 277082 is a ACAT-catalyzed cholesterol esterification and cholesterol absorption inhibitor .
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Cat. No.: HY-101576
CAS No.: 136609-26-2
Purity:  99.22%
Target:  

Acyltransferase

Research Areas:  

Metabolic Disease

RP 70676 is a potent inhibitor of ACAT, with IC50 of 25 and 44 nM for rat and rabbit ACAT.
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Cat. No.: HY-100288
CAS No.: 136609-53-5
Target:  

Acyltransferase

Research Areas:  

Metabolic Disease

RP 73163 Racemate is the racemate of RP 73163. RP 73163 is a potent ACAT inhibitor, with cholesterol lowering activity.
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Cat. No.: HY-N6702
CAS No.: 2503-13-1
Enniatin A is a Fusarium mycotoxin. Enniatin A inhibits acyl-CoA: cholesterol acyltransferase (ACAT) activity with an IC50 of 22 μM in an enzyme assay using rat liver microsomes .
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Cat. No.: HY-16281
CAS No.: 130804-35-2
Synonyms: DuP 128
Target:  

Acyltransferase

Research Areas:  

Metabolic Disease

Lecimibide (DuP 128) is a potent and specific acyl-CoA:cholesterol acyltransferase (ACAT) inhibitor for antihyperlipidemia research .
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Cat. No.: HY-139020
CAS No.: 454203-25-9
Target:  

Acyltransferase

Research Areas:  

Inflammation/Immunology

ACAT-IN-3 is an acyl-Coenzyme A:cholesterol acyltransferase (ACAT) inhibitor. ACAT-IN-3 inhibits NF-κB mediated transcription .
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Cat. No.: HY-139024
CAS No.: 199984-38-8
Target:  

Acyltransferase

Research Areas:  

Inflammation/Immunology

ACAT-IN-7 is an acyl-Coenzyme A:cholesterol acyltransferase (ACAT) inhibitor. ACAT-IN-7 inhibits NF-κB mediated transcription .
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Cat. No.: HY-139021
CAS No.: 454203-56-6
Target:  

Acyltransferase

Research Areas:  

Inflammation/Immunology

ACAT-IN-4 (Example 208) is an acyl-Coenzyme A:cholesterol acyltransferase (ACAT) inhibitor. ACAT-IN-4 inhibits NF-κB mediated transcription .
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Cat. No.: HY-139021A
CAS No.: 199984-46-8
Target:  

Acyltransferase

Research Areas:  

Inflammation/Immunology

ACAT-IN-4 hydrochloride (Example 208) is an acyl-Coenzyme A:cholesterol acyltransferase (ACAT) inhibitor. ACAT-IN-4 hydrochloride inhibits NF-κB mediated transcription .
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Cat. No.: HY-139022
CAS No.: 199983-93-2
Target:  

Acyltransferase

Research Areas:  

Inflammation/Immunology

ACAT-IN-5 (example 19) is an acyl-Coenzyme A:cholesterol acyltransferase (ACAT) inhibitor. ACAT-IN-5 inhibits NF-κB mediated transcription .
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Cat. No.: HY-139025
CAS No.: 199984-35-5
Target:  

Acyltransferase

Research Areas:  

Inflammation/Immunology

ACAT-IN-8 (example 206) is an acyl-Coenzyme A:cholesterol acyltransferase (ACAT) inhibitor. ACAT-IN-8 inhibits NF-κB mediated transcription .
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Cat. No.: HY-139019
CAS No.: 199984-55-9
Target:  

Acyltransferase

Research Areas:  

Inflammation/Immunology

ACAT-IN-2 is an acyl-Coenzyme A:cholesterol acyltransferase (ACAT) inhibitor extracted from patent EP1236468A1, example 187. ACAT-IN-2 inhibits NF-κB mediated transcription .
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Cat. No.: HY-139026
CAS No.: 199984-40-2
Target:  

Acyltransferase

Research Areas:  

Inflammation/Immunology

ACAT-IN-9 is an acyl-Coenzyme A:cholesterol acyltransferase (ACAT) inhibitor extracted from patent EP1236468A1, example 207. ACAT-IN-9 inhibits NF-κB mediated transcription .
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Cat. No.: HY-139023
CAS No.: 454203-45-3
Target:  

Acyltransferase

Research Areas:  

Inflammation/Immunology

ACAT-IN-6 is an acyl-Coenzyme A:cholesterol acyltransferase (ACAT) inhibitor extracted from patent EP1236468A1, example 200. ACAT-IN-6 potently inhibits NF-κB mediated transcription .
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Cat. No.: HY-139027
CAS No.: 454203-40-8
Target:  

Acyltransferase

Research Areas:  

Inflammation/Immunology

ACAT-IN-10 is an acyl-Coenzyme A:cholesterol acyltransferase (ACAT) inhibitor extracted from patent EP1236468A1, example 197. ACAT-IN-10 weakly inhibits NF-κB mediated transcription .
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Cat. No.: HY-139027A
CAS No.: 199983-77-2
Target:  

Acyltransferase

Research Areas:  

Inflammation/Immunology

ACAT-IN-10 dihydrochloride is an acyl-Coenzyme A:cholesterol acyltransferase (ACAT) inhibitor extracted from patent EP1236468A1, example 197. ACAT-IN-10 dihydrochloride weakly inhibits NF-κB mediated transcription .
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