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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
141 Results for "
Configuration
" in MedChemExpress (MCE) Product Catalog:
Products (141)
141 Results for "Configuration" in MCE Product Catalog:
Target:
Áreas de investigación:
SRI 6409-94 is an orally active Ro 13-6298 analogue that is teratogenic. SRI 6409-94 serves as a molecular tool to study the effect of the three-dimensional configuration of retinol on teratogenic activity .
Referencia número: HY-W010347R
No. CAS: 6027-13-0
Referencia número: HY-W012885
No. CAS: 53562-86-0
Áreas de investigación:
L-Inosine is the L-configuration of Inosine (HY-N0092). Inosine is an endogenous purine nucleoside produced by catabolism of adenosine .
Target:
Áreas de investigación:
(Z)-Lanoconazole is the Z configuration of Lanoconazole. Lanoconazole is a potent and orally active imidazole antifungal agent, shows a broad spectrum of activity against fungi in vitro and in vivo . Lanoconazole interferes with ergosterol biosynthesis by inhibiting sterol 14-alpha demethylase and blocking fungal membrane ergosterol biosynthesis. Lanoconazole can be used for the investigation of dermatophytosis and onychomycosis .
Referencia número: HY-W740611
No. CAS: 547-96-6
Category:
Target:
Referencia número: HY-B0196B
No. CAS: 93413-44-6
Target:
Áreas de investigación:
(S)-Venlafaxine is the (S)-configuration of Venlafaxine. Venlafaxine is an orally active, potent serotonin (5-HT)/norepinephrine (NE) reuptake dual inhibitor. Venlafaxine is an antidepressant agent .
Referencia número: HY-W160625
No. CAS: 1123-09-7
Target:
Referencia número: HY-177712
No. CAS: 1599530-54-7
Target:
Áreas de investigación:
RORγt inverse agonist 36 (S configuration of Compound 16) is a RORγt inverse agonist. RORγt inverse agonist 36 can be used for the research of inflammation and immunology .
Referencia número: HY-10082A
No. CAS: 200933-27-3
Synonyms: (E)-PAN-811; (E)-NSC# 663249; (E)-OCX191
Target:
Áreas de investigación:
(E)-3-AP is the E configuration of 3-AP. 3-AP is a potent ribonucleotide reductase inhibitor. 3-AP shows anti-proliferative activity. 3-AP shows anticancer activity in L1210 leukemia model. 3-AP inhibits RR activity and DNA synthesis .
Referencia número: HY-W856375
No. CAS: 953792-48-8
Referencia número: HY-122359A
No. CAS: 31477-60-8
Synonyms: rel-L-Centchroman; Ormeloxifene
Áreas de investigación:
rel-Levormeloxifene (rel-L-Centchroman) is the relative configuration of Levormeloxifene (HY-122359). rel-Levormeloxifene is a selective estrogen receptor modulator (SERM). rel-Levormeloxifene inhibits proliferation of leukemia cells with IC50 about 7 μM, arrests cell cycle at G0/G1 phase, and induces apoptosis. rel-Levormeloxifene induces differentation of myelogenesis leukemia, and enhances ROS production in K562 cells .
Referencia número: HY-101960
No. CAS: 122520-90-5
Synonyms: (Z)-AG-183
(Z)-Tyrphostin A51 is the Z configuration of Lanoconazole A51. Tyrphostin A51 is a potent protein tyrosine kinase (PTK) inhibitor. Tyrphostin A51 inhibits the volume-dependent release of [ 3H]taurine in a dose-dependent manner. Tyrphostin A51 markedly reduces cellular tyrosyl phosphorylation level. Tyrphostin A51 inhibits both basal and EGF-induced human bone cell proliferation .
Target:
Referencia número: HY-125949
No. CAS: 1445952-33-9
Target:
Referencia número: HY-106841A
No. CAS: 138681-29-5
Synonyms: (-)-Draflazine; (S)-R-75231; (S)-R88021
Target:
Áreas de investigación:
(S)-Draflazine ((-)-Draflazine) is the (S)-configuration of Draflazine (HY-106841). (S)-Draflazine is a potent blocker of nucleoside transport .
Referencia número: HY-W098280
No. CAS: 26682-99-5
Target:
Áreas de investigación:
Phenylglycine methyl ester is a chiral anisotropic reagent. Phenylglycine methyl ester can be used for absolute configuration determination of various chiral carboxylic acids .
Referencia número: HY-109092A
No. CAS: 2730989-98-5
Synonyms: rel-LIK066
Target:
Áreas de investigación:
rel-Licogliflozin is a relative configuration of Licogliflozin (HY-109092). Licogliflozin is a sodium glucose cotransporter (SGLT1 and SGLT2) inhibitor .
Referencia número: HY-P3045
No. CAS: 2393866-06-1
Target:
Áreas de investigación:
Referencia número: HY-125644
No. CAS: 18416-85-8
Target:
Áreas de investigación:
L-Lombricine is a D-configuration amino acid, which can be isolated from Lumbricus terrestris. L-Lombricine is related to the energy storage in earthworms .
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Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
