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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
76 Results for "
Epimer.
" in MedChemExpress (MCE) Product Catalog:
Products (76)
76 Results for "Epimer." in MCE Product Catalog:
Cat. No.: HY-129922
CAS No.: 773825-80-2
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Prostaglandin I2 is an unstable prostanoid which, through the ‘I prostanoid’ (IP) receptor, inhibits platelet aggregation and promotes vasodilatation in pulmonary vascular beds. AFP 07 is a 7,7-difluoroprostacyclin derivative that acts as a selective and highly potent agonist for the IP receptor (Ki=0.561 nM).1 AFP 07 shows weaker affinity for EP receptors, with Ki values > 100 nM for EP1-3 and > 10 nM for EP4. 16(R)-AFP 07 is an epimer of AFP 07. Its biological properties, particularly through the IP and EP receptors, remain to be evaluated.
Cat. No.: HY-125527AS
Synonyms: 17(R)-RvD1-d5; AT-RvD1-d5
Cat. No.: HY-Z19587
Synonyms: Ascomycin 19-epimer
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Tacrolimus impurity 3 (Ascomycin 19-epimer) is an impurity of Tacrolimus.
Cat. No.: HY-186146A
CAS No.: 3013618-85-1
Synonyms: SGI-1776-cis-VHL-02
SGI-1776-VHL-02-epimer (SGI-1776-cis-VHL-02) is an epimer control compound of with SGI-1776-VHL-02 (HY-186146). SGI-1776-VHL-02-epimer has an inverted stereocenter in the critical hydroxyl-proline group in the VHL ligand. SGI-1776-VHL-02-epimer cannot trigger the VHL E3 ligase complex and does not degrade PIM1 .
Cat. No.: HY-N21851
CAS No.: 145867-19-2
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Cat. No.: HY-N21698
CAS No.: 1253206-38-0
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Cat. No.: HY-N0210S5
CAS No.: 64267-73-8
Synonyms: D-(+)-Galactose-d1
Cat. No.: HY-161993A
CAS No.: 3043939-19-8
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(αR)-BI-9787 is the epimer of BI-9787 (HY-161993). BI-9787 is a zwitterionic inhibitior for ketohexokinase.
Cat. No.: HY-159465A
CAS No.: 2725913-38-0
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(S)-E3 ligase Ligand 30 is an E3 ligand that can be used for the synthesis of PROTACs, such as PRT3789 epimer (HY-159607A) .
Cat. No.: HY-172738A
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(S)-E3 Ligase Ligand-linker Conjugate 175 is a conjugate of an E3 ligase ligand and linker, which can be used for the synthesis of PROTACs, such as PRT3789 epimer (HY-159607A) .
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Phenindamine hydrochloride (Nu 1504 hydrochloride) is the hydrochloride salt of Phenindamine (HY-A0149). Phenindamine is a histamine H1 receptor antagonist. Phenindamine hydrochloride mainly exists in the 9-9a ene configuration and as a mixture of protonated epimers. Phenindamine hydrochloride can be used in studies related to histamine H1 receptor antagonists and the salt-type structure of Phenindamine .
Cat. No.: HY-172574
Synonyms: 8-iso-17-Phenyl trinor PGF2α
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8-Iso-17-phenyl trinor prostaglandin F2α (8-Iso-17-phenyl trinor PGF2), the C-8 epimer of Bimatoprost (HY-B0191), is a PGF2α (HY-12956) analog. Bimatoprost can be used in the research of glaucoma and high intraocular pressure.
Cat. No.: HY-182460
CAS No.: 173792-67-1
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Cat. No.: HY-W723158
CAS No.: 100992-60-7
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Epibestatin hydrochloride is an epimer of Bestatin (HY-B0134), a DPP4 inhibitor and protease inhibitor, with an IC50 of 17 μM against DPP4. As a stabilizer, Epibestatin hydrochloride binds to the cleft between 14-3-3 protein and plant proton pump PMA2, selectively stabilizing their interaction without affecting other 14-3-3 client proteins. Epibestatin hydrochloride triggers stomatal opening in leaf epidermis of Commelina communis. Epibestatin hydrochloride can be used in studies related to type 2 diabetes .
Cat. No.: HY-117580S2
Synonyms: OH-PRED-d5
Cat. No.: HY-145474
CAS No.: 937738-64-2
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17(R)-Resolvin D1 methyl ester is the methyl ester of Resolvin D1 (RvD1) (HY-125527) induced by Aspirin (HY-14654) with the 17R epimer (AT-RvD1). RvD is a regulator of transendothelial migration of human polymorphonuclear leukocytes and an anti-inflammatory agent. The 17R-trihydroxy-4Z of RvD1 also blocks transendothelial migration of human neutrophils (EC50 approximately 30 nM). AT-RvD1 is an effective form that protects against the rapid inactivation of Resolvin D1 .
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Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
