2 Results for "

4-OHT

" in MedChemExpress (MCE) Product Catalog:
Products (2)

2 Results for "4-OHT" in MCE Product Catalog:

3
(E/Z)-4-Hydroxytamoxifen
(E/Z)-4-Hydroxytamoxifen
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3 Cited Publications
Cat. No.: HY-16950A
CAS No.: 68392-35-8
Synonyms: Afimoxifene; 4-OHT
Category:  

Alkaloids Monophenols Other Alkaloids Phenols Endogenous metabolite Disease Research Fields Cancer

Target:  

Estrogen Receptor/ERR Adhesion G Protein-coupled Receptors (AGPCRs) Drug Metabolite

(E/Z)-4-Hydroxytamoxifen (Afimoxifene) is a racemic compound of (Z)-4-Hydroxytamoxifen and (E)-4-Hydroxytamoxifen isomers. (E/Z)-4-Hydroxytamoxifen is a selective estrogen receptor modulator with mixed estrogenic and antiestrogenic activity, which is also an active metabolite of Tamoxifen (HY-13757A). (E/Z)-4-Hydroxytamoxifen is an agonist of the G protein-coupled estrogen receptor (GPER) with relatively low affinity (100-1000 nM). (E/Z)-4-Hydroxytamoxifen is promising for research of cyclical mastalgia, such as breast pain, tenderness, and nodularity [4].
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(E/Z)-4-Hydroxytamoxifen (Standard)
(E/Z)-4-Hydroxytamoxifen (Standard)
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Cat. No.: HY-16950AR
CAS No.: 68392-35-8
Synonyms: Afimoxifene (Standard); 4-OHT (Standard)
Category:  

Alkaloids Monophenols Other Alkaloids Phenols Endogenous metabolite

Target:  

Reference Standards Estrogen Receptor/ERR Endogenous Metabolite

(E/Z)-4-Hydroxytamoxifen (Standard) is the analytical standard of (E/Z)-4-Hydroxytamoxifen. This product is intended for research and analytical applications. (E/Z)-4-Hydroxytamoxifen (Afimoxifene) is a racemic compound of (Z)-4-Hydroxytamoxifen and (E)-4-Hydroxytamoxifen isomers. (E/Z)-4-Hydroxytamoxifen is a selective estrogen receptor modulator with mixed estrogenic and antiestrogenic activity, which is also an active metabolite of Tamoxifen (HY-13757A). (E/Z)-4-Hydroxytamoxifen is an agonist of the G protein-coupled estrogen receptor (GPER) with relatively low affinity (100-1000 nM). (E/Z)-4-Hydroxytamoxifen is promising for research of cyclical mastalgia, such as breast pain, tenderness, and nodularity [4].
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