2 Results for "

CADA

" in MedChemExpress (MCE) Product Catalog:
Products (2)

2 Results for "CADA" in MCE Product Catalog:

Cat. No.: HY-134809
CAS No.: 182316-44-5
Purity:  98.45%
Synonyms: CADA
Target:  

HIV

Research Areas:  

Infection Inflammation/Immunology

Cyclotriazadisulfonamide (CADA) is a specific CD4-targeted HIV entry inhibitors. Cyclotriazadisulfonamide (CADA) inhibits the co-translational translocation of human CD4 (huCD4) into the ER lumen in a signal peptide (SP)-dependent way. Cyclotriazadisulfonamide is also a Sec61 translocon inhibitor .
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Cat. No.: HY-134809A
CAS No.: 392287-03-5
Synonyms: CADA hydrochloride
Target:  

HIV

Research Areas:  

Infection

Cyclotriazadisulfonamide (CADA) hydrochloride is a specific CD4-targeted HIV entry inhibitor with activity against HIV-1 replication. Cyclotriazadisulfonamide hydrochloride can specifically downregulate the expression of CD4 receptors on the cell surface, effectively inhibiting HIV transmission. Cyclotriazadisulfonamide hydrochloride can inhibit HIV-1(NL4.3) and SIV(mac251), and has a synergistic effect when used in combination with cellulose acetate (CAP). Cyclotriazadisulfonamide hydrochloride can also be used as a microbial gel formulation to maintain CD4 downregulation and antiviral activity, and is a broad-spectrum anti-HIV agent.
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