2 Results for "

CCG50014

" in MedChemExpress (MCE) Product Catalog:
Products (2)

2 Results for "CCG50014" in MCE Product Catalog:

2
2 Cited Publications
Cat. No.: HY-13509
CAS No.: 883050-24-6
Purity:  99.62%
Target:  

RGS Protein

Research Areas:  

Inflammation/Immunology

CCG-50014 is the most potent against the regulator of G-protein signaling protein type 4 (RGS4) (IC50 =30 nM) and is >20-fold selective for RGS4 over other RGS proteins. CCG-50014 binds covalently to the RGS, forming an adduct on two cysteine residues located in an allosteric regulatory site . CCG50014, reduces nociceptive responses and enhances opioid-mediated analgesic effects in the mouse formalin test .
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Cat. No.: HY-13509R
CAS No.: 883050-24-6
Target:  

RGS Protein

Research Areas:  

Inflammation/Immunology

CCG-50014 (Standard) is the analytical standard of CCG-50014. This product is intended for research and analytical applications. CCG-50014 is the most potent against the regulator of G-protein signaling protein type 4 (RGS4) (IC50 =30 nM) and is >20-fold selective for RGS4 over other RGS proteins. CCG-50014 binds covalently to the RGS, forming an adduct on two cysteine residues located in an allosteric regulatory site . CCG50014, reduces nociceptive responses and enhances opioid-mediated analgesic effects in the mouse formalin test .
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