1 Result for "

CTEP

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "CTEP" in MCE Product Catalog:

2
2 Cited Publications
Referencia número: HY-15445
No. CAS: 871362-31-1
Pureza:  99.59%
Synonyms: RO 4956371; mGluR5 inhibitor
Target:  

mGluR

Áreas de investigación:  

Neurological Disease

CTEP (RO 4956371) is a novel, long-acting, orally bioavailable allosteric antagonist of mGlu5 receptor with IC50 of 2.2 nM, and shows > 1000-fold selectivity over other mGlu receptors. CTEP is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.
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