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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
6 Results for "
Defactinib
" in MedChemExpress (MCE) Product Catalog:
Products (6)
6 Results for "Defactinib" in MCE Product Catalog:
59
59 Cited Publications
Synonyms: VS-6063; PF-04554878
Defactinib (VS-6063; PF-04554878) is a novel FAK inhibitor with potential antiangiogenic and antineoplastic activities.
59
59 Cited Publications
Synonyms: VS-6063 hydrochloride; PF 04554878 hydrochloride
Defactinib hydrochloride (VS-6063 hydrochloride; PF 04554878 hydrochloride) is a novel FAK inhibitor, which inhibits FAK phosphorylation at the Tyr397 site in a time- and dose-dependent manner.
Cat. No.: HY-12289R
CAS No.: 1073154-85-4
Synonyms: VS-6063 (Standard); PF-04554878 (Standard)
Target:
Research Areas:
Defactinib (Standard) is the analytical standard of Defactinib. This product is intended for research and analytical applications. Defactinib (VS-6063; PF-04554878) is a novel FAK inhibitor with potential antiangiogenic and antineoplastic activities.
Cat. No.: HY-12289S
CAS No.: 2384121-03-1
Synonyms: VS-6063-d6; PF-04554878-d6
Cat. No.: HY-12289AR
CAS No.: 1073160-26-5
Synonyms: VS-6063 hydrochloride (Standard); PF 04554878 hydrochloride (Standard)
Target:
Research Areas:
Defactinib (hydrochloride) (Standard) is the analytical standard of Defactinib (hydrochloride). This product is intended for research and analytical applications. Defactinib hydrochloride (VS-6063 hydrochloride; PF 04554878 hydrochloride) is a novel FAK inhibitor, which inhibits FAK phosphorylation at the Tyr397 site in a time- and dose-dependent manner.
Cat. No.: HY-44146
CAS No.: 2296719-34-9
Research Areas:
Defactinib analogue-1 (Compound 7) is a ligand for target protein Fak, that can be used for synthesis of PROTAC FAK degrader 1 (HY-119932) .
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Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
