7 Results for "

Eletriptan

" in MedChemExpress (MCE) Product Catalog:
Products (7)

7 Results for "Eletriptan" in MCE Product Catalog:

1
1 Cited Publications
Cat. No.: HY-A0010
CAS No.: 177834-92-3
Synonyms: Eletriptan HBr; UK-116044 hydrobromide
Target:  

5-HT Receptor

Research Areas:  

Neurological Disease

Eletriptan hydrobromide (Eletriptan HBr) is a 5-HT1B and 5-HT1D receptor agonist with antimigraine activity, with Ki of 0.92 nM and 3.14 nM, respectively .
loading...
    loading...
Cat. No.: HY-A0039S1
CAS No.: 1126745-65-0
Eletriptan-d5 is the deuterium labeled Eletriptan . Eletriptan (UK-116044) is a highly selective and orally active serotonin 5-HT1B and 5-HT1D receptor agonist, with pKi values of 8.0 and 8.9, respectively. Eletriptan has inhibitory effects on markers of neurogenic inflammation in rats. Eletriptan can be used for researching migraine .
loading...
    loading...
Cat. No.: HY-A0039
CAS No.: 143322-58-1
Synonyms: UK-116044
Eletriptan (UK-116044) is a highly selective and orally active serotonin 5-HT1B and 5-HT1D receptor agonist, with pKi values of 8.0 and 8.9, respectively. Eletriptan has inhibitory effects on markers of neurogenic inflammation in rats. Eletriptan can be used for researching migraine .
loading...
    loading...
Cat. No.: HY-137580
CAS No.: 153525-55-4
Target:  

Cytochrome P450

Research Areas:  

Metabolic Disease

N-desmethyl Eletriptan is a metabolite of Eletriptan (HY-A0039). It is formed from eletriptan primarily by the cytochrome P450 (CYP) isoform CYP3A4 in human liver microsomes.
loading...
    loading...
Cat. No.: HY-A0039S2
Eletriptan-d5 (hydrochloride) is the deuterium labeled Eletriptan hydrochloride . Eletriptan (UK-116044) hydrochloride is a highly selective and orally active serotonin 5-HT1B and 5-HT1D receptor agonist, with pKi values of 8.0 and 8.9, respectively. Eletriptan hydrochloride has inhibitory effects on markers of neurogenic inflammation in rats. Eletriptan hydrochloride can be used for researching migraine .
loading...
    loading...
Cat. No.: HY-A0010R
CAS No.: 177834-92-3
Synonyms: Eletriptan HBr (Standard); UK-116044 hydrobromide (Standard)
Research Areas:  

Neurological Disease

Eletriptan hydrobromide (Standard) is an analytical standard for Eletriptan hydrobromide. This product is intended for research and analytical applications. Eletriptan hydrobromide (Eletriptan HBr) is a 5-HT1B and 5-HT1D receptor agonist with antimigraine activity, with Ki of 0.92 nM and 3.14 nM, respectively .
loading...
    loading...
Cat. No.: HY-A0039S
CAS No.: 1287040-94-1
Synonyms: UK-116044-d3
Eletriptan-d3 is the deuterium labeled Eletriptan hydrobromide. Eletriptan hydrobromide is a selective 5-HT1B and 5-HT1D receptor agonist with Ki of 0.92 nM and 3.14 nM, respectively .
loading...
    loading...