3 Results for "

GEA654

" in MedChemExpress (MCE) Product Catalog:
Products (3)

3 Results for "GEA654" in MCE Product Catalog:

Cat. No.: HY-133732
CAS No.: 60719-83-7
Synonyms: GEA 654 hydrochloride; A03 hydrochloride
Alaproclate (GEA 654) hydrochloride is a selective and orally active serotonin re-uptake inhibitor (SSRI). Alaproclate hydrochloride also acts as a potent, reversible and noncompetitive antagonist of the NMDA receptor coupled ion flow .
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Cat. No.: HY-124779
CAS No.: 66171-75-3
Synonyms: (S)-GEA 654; (S)-A03
Target:  

iGluR

(S)-Alaproclate ((S)-GEA 654) is more potent than the R-(+)-enantiomer both in blocking the NMDA receptor currents in vitro and in antagonizing the cGMP increase in vivo .
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Cat. No.: HY-124779A
CAS No.: 57469-92-8
Synonyms: (S)-GEA 654 hydrochloride; (S)-A03 hydrochloride
Target:  

Serotonin Transporter

Research Areas:  

Neurological Disease

(S)-Alaproclate ((S)-A03) hydrochloride is a potent selective serotonin reuptake inhibitor (SSRI), which is used as an antidepressant agent. (S)-Alaproclate (hydrochloride) also produces a potent block of N-methyl-d-aspartate (NMDA) receptor currents in hippocampal neurons (IC50=1.1 μM) with a potent blocker of K + currents .
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