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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
3 Results for "
GSK866
" in MedChemExpress (MCE) Product Catalog:
Products (3)
3 Results for "GSK866" in MCE Product Catalog:
Synonyms: (S)-GSK47866A
Target:
Forschungsgebiete:
GSK866 ((S)-GSK47866A) is a selective glucocorticoid receptor agonist, with an IC50 of 4.6 nM .
Art. -Nr.: HY-157294B
CAS. Nr.: 960248-81-1
Synonyms: GSK47866A
Target:
Forschungsgebiete:
(Rac)-GSK866 (GSK47866A) is a non-steroidal glucocorticoid receptor (GR) ligand. The crystal structure of (Rac)-GSK866 bound to the GR LBD (3E7C) can be used as a model to study the mechanism of action of ligands of the same class .
Synonyms: (R)-GSK47866A
Target:
Forschungsgebiete:
(R)-GSK866 ((R)-GSK47866A) is the (R)-enantiomer of GSK866 (HY-157294). GSK866 is a selective agonist for glucocorticoid receptor with an IC50 of 4.6 nM .
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Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
