3 Results for "

Mavatrep

" in MedChemExpress (MCE) Product Catalog:
Products (3)

3 Results for "Mavatrep" in MCE Product Catalog:

Cat. No.: HY-16935
CAS No.: 956274-94-5
Synonyms: JNJ-39439335
Target:  

TRP Channel

Research Areas:  

Neurological Disease

Mavatrep (JNJ-39439335) is an orally active, selective and potent TRPV1 antagonist with high affinity for hTRPV1 channels (Ki=6.5 nM). Mavatrep antagonizes capsaicin-induced Ca 2+ influx with an IC50 value of 4.6 nM. Mavatrep can be used in some studies of neuropathic pain .
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Cat. No.: HY-16935S
Synonyms: JNJ-39439335-d6
Mavatrep-d6 (JNJ-39439335-d6) is a deuterated labeled Mavatrep (HY-16935). Mavatrep (JNJ-39439335) is an orally active, selective and potent TRPV1 antagonist with high affinity for hTRPV1 channels (Ki=6.5 nM). Mavatrep antagonizes capsaicin-induced Ca 2+ influx with an IC50 value of 4.6 nM. Mavatrep can be used in some studies of neuropathic pain .
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Cat. No.: HY-16935R
CAS No.: 956274-94-5
Synonyms: JNJ-39439335 (Standard)
Research Areas:  

Neurological Disease

Mavatrep (Standard) is the analytical standard of Mavatrep. This product is intended for research and analytical applications. Mavatrep (JNJ-39439335) is an orally active, selective and potent TRPV1 antagonist with high affinity for hTRPV1 channels (Ki=6.5 nM). Mavatrep antagonizes capsaicin-induced Ca2+ influx with an IC50 value of 4.6 nM. Mavatrep can be used in some studies of neuropathic pain .
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