4 Results for "

NO711

" in MedChemExpress (MCE) Product Catalog:
Products (4)

4 Results for "NO711" in MCE Product Catalog:

Cat. No.: HY-103506
CAS No.: 145645-62-1
Purity:  99.76%
Synonyms: NO-711 hydrochloride
Target:  

GABA Receptor

Research Areas:  

Neurological Disease

NNC-711 (NO-711 hydrochloride) is a potent and selective inhibitor of GAT-1 (GABA transporter 1) with IC50 values of 0.04, 0.38, 171, 1700, 349, 622 μM for human GAT-1, rat GAT-1, rGAT-2, hGAT-3, rGAT-3, hBGT-3, respectively. NNC-711 has anticonvulsant and analgesic effect in vivo and exhibits cognition-enhancing activity .
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Cat. No.: HY-114040
CAS No.: 159094-94-7
Synonyms: NNC-711 free acid
Target:  

GABA Receptor

Research Areas:  

Neurological Disease

NO-711 (NNC-711) free acid is a novel potent and selective inhibitor of γ-aminobutyric acid uptake. NO-711 inhibits synaptosomal (IC50 = 47 nM), neuronal (IC50 = 1238 nM) and glial (IC50 = 636 nM) GABA uptake in vitro .
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Cat. No.: HY-129464
CAS No.: 127586-66-7
Target:  

GABA Receptor

Research Areas:  

Neurological Disease

NO-711ME is a prodrug of NO-711. NO-711 is a potent and selective GABA uptake inhibitor .
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Cat. No.: HY-103506R
CAS No.: 145645-62-1
Synonyms: NO-711 hydrochloride (Standard)
Research Areas:  

Neurological Disease

NNC-711 (Standard) is the analytical standard of NNC-711 (HY-103506). This product is intended for research and analytical applications. NNC-711 (NO-711 hydrochloride) is a potent and selective inhibitor of GAT-1 (GABA transporter 1) with IC50 values of 0.04, 0.38, 171, 1700, 349, 622 μM for human GAT-1, rat GAT-1, rGAT-2, hGAT-3, rGAT-3, hBGT-3, respectively. NNC-711 has anticonvulsant and analgesic effect in vivo and exhibits cognition-enhancing activity .
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