1 Result for "

Q94

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "Q94" in MCE Product Catalog:

Cat. No.: HY-108554
CAS No.: 1052076-77-3
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Q94 hydrochloride, a selective PAR1 antagonist (IC50=916 nM), can selectively block PAR1/Gαq interaction and signalling. Q94 hydrochloride blocks PAR1-mediated increases in both CCL2 mRNA and protein levels in a dose-dependent manner. Q94 hydrochloride also completely blocks thrombin-induced ERK1/2 and MLC phosphorylation .
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