3 Results for "

TAK147

" in MedChemExpress (MCE) Product Catalog:
Products (3)

3 Results for "TAK147" in MCE Product Catalog:

Cat. No.: HY-19651A
CAS No.: 142852-51-5
Synonyms: TAK-147
Target:  

Cholinesterase (ChE)

Research Areas:  

Neurological Disease

Zanapezil (TAK-147) is a potent, reversible and selective acetylcholine esterase (AChE) inhibitor. Zanapezil shows a potent and reversible inhibition of AChE activity in homogenates of the rat cerebral cortex (IC50=51.2 nM). Zanapezil shows a moderate inhibition of muscarinic M1 and M2 receptor binding with Ki values of 234 and 340 nM, respectively. Zanapezil can be used for the research of early stages of Alzheimer's disease (AD) .
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Cat. No.: HY-19651B
CAS No.: 263248-42-6
Synonyms: TAK-147 fumarate
Target:  

Cholinesterase (ChE)

Research Areas:  

Neurological Disease

Zanapezil (TAK-147) fumarate is a potent, reversible and selective acetylcholine esterase (AChE) inhibitor. Zanapezil fumarate shows a potent and reversible inhibition of AChE activity in homogenates of the rat cerebral cortex (IC50=51.2 nM). Zanapezil fumarate shows a moderate inhibition of muscarinic M1 and M2 receptor binding with Ki values of 234 and 340 nM, respectively. Zanapezil fumarate can be used for the research of early stages of Alzheimer's disease (AD) .
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Cat. No.: HY-19651
CAS No.: 142852-50-4
Synonyms: TAK-147 free base
Target:  

Cholinesterase (ChE)

Research Areas:  

Neurological Disease

Zanapezil (TAK-147) free base is a potent, reversible and selective acetylcholine esterase (AChE) inhibitor. Zanapezil free base shows a potent and reversible inhibition of AChE activity in homogenates of the rat cerebral cortex (IC50=51.2 nM). Zanapezil free base shows a moderate inhibition of muscarinic M1 and M2 receptor binding with Ki values of 234 and 340 nM, respectively. Zanapezil free base can be used for the research of early stages of Alzheimer's disease (AD) .
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