5 Results for "

XL147

" in MedChemExpress (MCE) Product Catalog:
Products (5)

5 Results for "XL147" in MCE Product Catalog:

12
12 Publications Verification
Cat. No.: HY-12068
CAS No.: 1349796-36-6
Purity:  99.46%
Synonyms: XL-147 derivative 1
Target:  

PI3K

Research Areas:  

Cancer

PI3K-IN-1 (XL-147 derivative 1) is a potent inhibitor of PI3K. PI3K-IN-1 (25 μM) blocks PI3K/Akt signaling pathways .
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6
6 Cited Publications
Cat. No.: HY-16526
CAS No.: 934526-89-3
Synonyms: XL-147; SAR245408
Target:  

PI3K

Research Areas:  

Cancer

Pilaralisib (XL147; SAR245408) is a potent and highly selective class I PI3Ks inhibitor with IC50s of 39 nM, 383 nM, 23 nM and 36 nM for PI3Kα, PI3Kβ, PI3Kγ, and PI3Kδ.
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1
1 Cited Publications
Cat. No.: HY-11105
CAS No.: 956958-53-5
Purity:  99.74%
Synonyms: XL147 analogue
Target:  

PI3K Apoptosis

Research Areas:  

Cancer

Pilaralisib analogue (XL147 analogue) is a representative and selective PI3Kα inhibitor extracted from patent WO2012006552A1, Compound 147 in Table 1.
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Cat. No.: HY-16526R
CAS No.: 934526-89-3
Synonyms: XL-147 (Standard); SAR245408 (Standard)
Research Areas:  

Cancer

Pilaralisib (Standard) is the analytical standard of Pilaralisib. This product is intended for research and analytical applications. Pilaralisib (XL147; SAR245408) is a potent and highly selective class I PI3Ks inhibitor with IC50s of 39 nM, 383 nM, 23 nM and 36 nM for PI3Kα, PI3Kβ, PI3Kγ, and PI3Kδ.
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Cat. No.: HY-12068R
CAS No.: 1349796-36-6
Synonyms: XL-147 derivative 1 (Standard)
Research Areas:  

Cancer

PI3K-IN-1 (Standard) is the analytical standard of PI3K-IN-1. This product is intended for research and analytical applications. PI3K-IN-1 (XL-147 derivative 1) is a potent inhibitor of PI3K. PI3K-IN-1 (25 μM) blocks PI3K/Akt signaling pathways .
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