1 Result for "

guanidine-based

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "guanidine-based" in MCE Product Catalog:

Cat. No.: HY-12896
CAS No.: 1449765-65-4
Target:  

SphK

Research Areas:  

Cancer

SLR080811 is a guanidine-based selective sphingosine kinase 2 (SphK2) inhibitor with a Ki of 1.3 μM, exhibiting ~10-fold selectivity over SphK1 (Ki = 12 μM). SLR080811 reduces sphingosine 1-phosphate (S1P) levels in vitro, but drives a SphK1-dependent increase in S1P in mice. SLR080811 can be used for cancers and fibrosis research .
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