17β-HSD10-IN-1
Based on 1 Customer Validation
17β-HSD10-IN-1 (compound 9) is an orally active inhibitor of 17β-hydroxysteroid dehydrogenase type 10 (17β-HSD10) with blood-brain permeability. 17β-HSD10-IN-1 doesn't result additional effects for mitochondrial off-targets and cytotoxic or neurotoxic effects.
For research use only. We do not sell to patients.
- Purity: 97.16%
- CAS No.: 2316765-78-1
- Formula: C16H13ClN4O3S
- Molecular Weight:376.82
-
Storage:Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
-
Biological Activity
-
Chemical Information
-
Solvent & Solubility
- Purity & Documentation
- References
-
Help & FAQs
-
Metabolism/Protease Compound Library
HY-L012
-
Phenols Library
HY-L057
-
Orally Active Compound Library
HY-L061
-
Metabolic Enzyme Compound Library
HY-L146
-
Bioactive Compound Library Max
HY-L181
-
MCE Bioactive Compound Library
HY-L001V
-
Bioactive Compound Library
HY-L001
-
RO5 Drug-like Natural Product Library
HY-L200
-
High-Throughput Bioactive Compound Library
HY-L205
-
Natural Product Diversity Scaffold Library
HY-L245
All 17β-HSD Isoforms
More
Biological Activity
17β-HSD10[1]
Chemical Information
-
CAS No. 2316765-78-1
-
Appearance Solid
-
Molecular Weight 376.82
-
Formula C16H13ClN4O3S
-
Color Pale purple to purple
-
SMILES
O=C(NC1=CC=C(C(Cl)=C1)O)NC(SC2=C3)=NC2=CC=C3NC(C)=O
-
Structure Classification
-
Initial Source
-
Shipping
Room temperature in continental US; may vary elsewhere.
-
Storage
Powder -20°C 3 years 4°C 2 years In solvent -80°C 6 months -20°C 1 month
Solvent & Solubility
DMSO : 25 mg/mL (66.34 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Purity & Documentation
-
Data Sheet (270 KB)
-
SDS (252 KB)
- English - EN (252 KB)
- Français - FR (252 KB)
- Deutsch - DE (252 KB)
- Norwegian - NO (252 KB)
- Español - ES (252 KB)
- Swedish - SV (252 KB)
- Italian - IT (252 KB)
- Korean - KR (252 KB)
- Portuguese - PT (252 KB)
-
Handling Instructions (2659 KB)
References
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 2.6538 mL | 13.2689 mL | 26.5379 mL | 66.3447 mL |
| 5 mM | 0.5308 mL | 2.6538 mL | 5.3076 mL | 13.2689 mL | |
| 10 mM | 0.2654 mL | 1.3269 mL | 2.6538 mL | 6.6345 mL | |
| 15 mM | 0.1769 mL | 0.8846 mL | 1.7692 mL | 4.4230 mL | |
| 20 mM | 0.1327 mL | 0.6634 mL | 1.3269 mL | 3.3172 mL | |
| 25 mM | 0.1062 mL | 0.5308 mL | 1.0615 mL | 2.6538 mL | |
| 30 mM | 0.0885 mL | 0.4423 mL | 0.8846 mL | 2.2115 mL | |
| 40 mM | 0.0663 mL | 0.3317 mL | 0.6634 mL | 1.6586 mL | |
| 50 mM | 0.0531 mL | 0.2654 mL | 0.5308 mL | 1.3269 mL | |
| 60 mM | 0.0442 mL | 0.2211 mL | 0.4423 mL | 1.1057 mL |
17β-HSD10-IN-1 Related Classifications
HY-155534 Related Classifications
Powered by Bioz