5-HT2A receptor activator-1
5-HT2A receptor activator-1 is an allosteric modulator of the 5-HT2A receptor, with an EC50 of 0.56 μM. 5-HT2A receptor activator-1 exerts allosteric interaction with the 5-HT2A receptor, enhances 5-HT-induced receptor activation by binding to the allosteric site, and shows no obvious agonistic activity on its own. 5-HT2A receptor activator-1 can be used in the research of neurological or psychiatric disorders.
For research use only. We do not sell to patients.
- CAS No.: 3129083-72-0
- Formula: C26H22F2N2O2S
- Molecular Weight:464.53
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
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- References
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Biological Activity
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5-HT2A Receptor 0.56 μM (EC50) |
5-HT2A receptor activator-1 (compound 5) (up to 10 μM; 50 min) acts as a positive allosteric modulator of human 5-HT2A receptor-expressing cells, with an EC50 of 0.56 μM and an Emax of 73%, and exhibits no orthosteric agonist activity at concentrations up to 10 μM[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 3129083-72-0
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Molecular Weight 464.53
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Formula C26H22F2N2O2S
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SMILES
O=S(C1=CC=C(C2=CC=C(F)C=C2)C=C1)(C)=NC3=CC=C(C(F)=C3)OC4=CC(C)=NC(C)=C4
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
5-HT2A receptor activator-1 Related Classifications
HY-187504 Related Classifications
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