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Cat. No.: HY-168334

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5-HT2C agonist-4

5-HT2C agonist-4 (Compound 3i) is an agonist for 5-HT2C receptor with an EC₅₀ of 5.7 nM. 5-HT2C agonist-4 reduces locomotor activity in the zebrafish larval model.

For research use only. We do not sell to patients.

CAS No.: 2730085-33-1
Formula: C₂₄H₂₅N₅O
Molecular Weight:399.49

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (273 KB)

5-HT2C agonist-4 Chemical Structure

CAS No.: 2730085-33-1

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Use of MCE Products

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity
- Description
- IC₅₀ & Target
Chemical Information
Purity & Documentation
References
Calculators
Help & FAQs
Classifications
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Biological Activity

Description

5-HT2C agonist-4 (Compound 3i) is an agonist for 5-HT2C receptor with an EC₅₀ of 5.7 nM. 5-HT2C agonist-4 reduces locomotor activity in the zebrafish larval model^[1].

IC₅₀ & Target

5-HT_2C Receptor

5.7 nM (EC₅₀)

5-HT_2A Receptor

139.4 nM (EC₅₀)

5-HT_2B Receptor

852 nM (EC₅₀)

All 5-HT Receptor Isoforms :

Chemical Information

CAS No. 2730085-33-1
Molecular Weight 399.49
Formula C₂₄H₂₅N₅O
SMILES

O=C(C1=C(/N=C/C2=CN(CC3=CC=CC=C3)C4=C2C=CC=C4)C(CCC)=NN1C)N
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (273 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

References

[1]. Reddy GS, et al., Amberlyst-15 catalysed synthesis of novel indole derivatives under ultrasound irradiation: Their evaluation as serotonin 5-HT2C receptor agonists. Bioorg Chem. 2021 Nov;116:105380. [Content Brief]

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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100 mg

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Biological Activity
- Description
- IC₅₀ & Target
Chemical Information
Purity & Documentation
References

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5-HT2C agonist-4

All 5-HT Receptor Isoforms