1. Signaling Pathways
  2. Metabolic Enzyme/Protease
  3. Dipeptidyl Peptidase
  4. DPP-4 Isoform
  5. DPP-4 Inhibitor

DPP-4 Inhibitor

DPP-4 Inhibitors (11):

Cat. No. Product Name Effect Purity
  • HY-14877
    Anagliptin
    Inhibitor
    Anagliptin (SK-0403) is a highly selective, potent, orally active inhibitor of dipeptidyl peptidase 4 (DPP-4), with an IC50 of 3.8 nM, and less selective at DPP-8 and DDP-9 with IC50s of 68 nM and 60 nM, respectively.
  • HY-13749A
    Sitagliptin phosphate
    Inhibitor 99.98%
    Sitagliptin phosphate (MK-0431 phosphate) is a potent inhibitor of DPP4 with an IC50 of 19 nM in Caco-2 cell extracts.
  • HY-117985B
    Evogliptin tartrate
    Inhibitor 99.96%
    Evogliptin (DA-1229) tartrate is an orally active DPP4 inhibitor with significant and sustained hypoglycaemic effects in mouse models.
  • HY-147401
    Sitagliptin fenilalanil
    Inhibitor
    Sitagliptin fenilalanil is a dipeptidyl aminopeptidase 4 (DPP-4) inhibitor.
  • HY-14877A
    Anagliptin hydrochloride
    Inhibitor
    Anagliptin (SK-0403) hydrochloride is a highly selective, potent, orally active inhibitor of dipeptidyl peptidase 4 (DPP-4), with an IC50 of 3.8 nM, and less selective at DPP-8 and DDP-9 with IC50s of 68 nM and 60 nM, respectively.
  • HY-151383
    DPP-4-IN-1
    Inhibitor
    DPP-4-IN-1 (compound d1) is a potent DPP-4 (dipeptidyl peptidase 4) inhibitor, with an IC50of 49 nM.
  • HY-151384
    DPP-4-IN-2
    Inhibitor
    DPP-4-IN-2 (compound b2) is a potent DPP-4 (dipeptidyl peptidase 4) inhibitor, with an IC50of 79 nM.
  • HY-13749C
    (S)-Sitagliptin phosphate
    Inhibitor
    (S)-Sitagliptin phosphate is the less active S-enantiomer of Sitagliptin phosphate.
  • HY-146455
    DPP-4-IN-3
    Inhibitor
    DPP-4-IN-3 (Compound 5a) is a potent dipeptidyl peptidase IV (DPP-IV) inhibitor with an IC50 of 0.75 nM.
  • HY-14806S
    Teneligliptin-d8
    Inhibitor
    Teneligliptin D8 (MP-513 D8) a deuterium labeled Teneligliptin (MP-513).
  • HY-129736
    P32/98 hemifumarate
    Inhibitor
    P32/98 hemifumarateis a potent inhibitor of dipeptidyl peptidase IV with a Ki value of 130 nM.