1. Signaling Pathways
  2. Immunology/Inflammation
  3. SphK
  4. SphK Inhibitors

SphK Inhibitors

SphK1

SphK2

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

SphK Inhibitors & Activators
Product Name SphK1 SphK2 Purity
PF-543
SphK1
  99.85%
PF-543 Citrate
SphK1
  99.47%
SLR080811
SphK1, Ki: 12 μM
SphK2, Ki: 1.3 μM
(R)-FTY720-OMe  
SphK2, IC50: 16.5 μM
K145 hydrochloride  
SphK2
99.63%
K6PC-5
SphK1
  99.27%
SK1-I
SphK1
  98.83%
SKI-178
SphK1
SphK2
99.29%
MP-A08
SphK1
  98.0%
MHP
SphK1
  98.57%
SK1-IN-1
SphK1
  98.10%
Amgen-23
SphK1, IC50: 20 nM
SphK2, IC50: 1.6 μM
98.11%
SphK1&2-IN-1
SphK1
SphK2
98.47%
SLM6031434 hydrochloride
SphK1, IC50: 16 μM
SphK2, IC50: 0.4 μM
99.1%
SphK2-IN-1  
SphK2, IC50: 0.359 μM
99.61%
CAY10621
SphK1
  99.3%
SLP7111228 hydrochloride
SphK1
  98.01%
PF-543 hydrochloride
SphK1
 
SphK1-IN-2
SphK1, IC50: 19.81 nM
SphK2, IC50: >10 μM
SLM6031434
SphK1, IC50: 16 μM
SphK2, IC50: 0.4 μM
SphK1-IN-4
SphK1
 
SphK1-IN-1
SphK1
 
SLP7111228
SphK1
 
ABC294735
SphK1
SphK2
SphK2-IN-4  
SphK2
VT-ME6  
SphK2, Ki: 8 μM
SphK1-IN-3
SphK1, IC50: 2.48 μM
 
RB-005
SphK1, IC50: 3.6 μM