1. Signaling Pathways
  2. JAK/STAT Signaling
    Stem Cell/Wnt
  3. STAT
  4. STAT Inhibitors

STAT Inhibitors

STAT3

STAT5

STAT6

STAT1

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STAT Inhibitors, Agonists, Antagonists, Activators, Modulators, Inducers, Degraders & Ligands
Product Name STAT3 STAT5 STAT6 STAT1 Purity
Sorafenib
STAT3
      99.85%
Stattic
STAT3
      99.96%
Cilengitide
STAT3 ([3])
      99.91%
Artesunate
Stat-3
      99.89%
STAT6-IN-10    
STAT6, EC50: 0.002 μM
  98.81%
GYY4137
Stat-3
      98.08%
Homoharringtonine
STAT3
      99.96%
AS1517499    
STAT6, IC50: 21 nM
  99.17%
Niclosamide
STAT3, IC50: 0.25 μM (in HeLa cells)
      99.96%
AG490
Stat-3
      99.86%
C188-9
STAT3, Kd: 4.7 nM
      99.84%
Colivelin
STAT3
      99.92%
TPCA-1
STAT3
      99.66%
NSC 74859
STAT3, IC50: 86 μM
      98.35%
Ritlecitinib
STAT3
STAT5
STAT6
  99.80%
Astaxanthin
STAT3
      98.0%
Scutellarin
STAT3
      99.57%
WP1066
STAT3
      99.77%
Cryptotanshinone
STAT3, IC50: 4.6 μM
      99.07%
Napabucasin
STAT3
      99.94%
Butyzamide
STAT3
STAT5
    99.83%
STAT5-IN-1  
STAT5β, IC50: 47 μM
    98.35%
Pimozide
STAT3
STAT5
    99.94%
AK-1690    
STAT6, DC50: 1 nM
  99.91%
Gamma-glutamylcysteine    
STAT6
  98.53%
SD-36
STAT3, Kd: 50 nM
      99.73%
Diosgenin
STAT3
      99.92%
KT-333
STAT3
      98.91%
Sorafenib tosylate
STAT3
      99.98%
AC-4-130  
STAT5
    99.93%
Saikosaponin D
STAT3
      99.81%
2-Chloro-5-(trifluoromethyl)pyrimidine      
STAT1
99.96%
AS2863619  
STAT5
    98.02%
Colivelin TFA
STAT3
      99.79%
1-Stearoyl-sn-glycero-3-phosphocholine
p-STAT3
      99.53%
SC-43
p-STAT3
      99.01%
AK-2292  
STAT5, DC50: 0.10 μM
    99.73%
Morusin
STAT3
      99.54%
SI-109
STAT3, Ki: 9 nM
      99.91%
ML115
Stat-3, EC50: 2 nM
      99.98%
Cucurbitacin I
STAT3
      99.56%
BP-1-102
STAT3, IC50: 6.8 μM
      99.26%
SH-4-54
STAT3, Kd: 300 nM
STAT5, Kd: 464 nM
    99.80%
Anti-Mouse NK1.1 Antibody (PK136)
p-STAT3
   
STAT1
98.57%
Anti-IL11 Antibody (X203)
STAT3
      98.53%
Erasin
STAT3, IC50: 9.7 μM
   
STAT1, IC50: 24 μM
YM-341619    
STAT6, IC50: 0.70 nM
  98.01%
STAT3-IN-1
Stat-3, IC50: 1.82 μM (in HT29 cells)
Stat-3, IC50: 2.14 μM (in MDA-MB 231 cells)
     
Alantolactone
STAT3
      99.94%
Guanosine 5'-diphosphate sodium, 96% (HPLC)
Stat-3
      99.88%
Stapokibart    
STAT6
  99.37%
Anti-Mouse IL-6 Antibody (MP5-20F3)
STAT3
      99.36%
BCI-137      
STAT1
99.84%
STAT6-IN-5    
STAT6, IC50: 0.24 μM
  99.88%
STAT6-IN-4    
STAT6, IC50: 0.34 μM
  99.77%
Nifuroxazide
STAT3
      99.90%
Perindopril
STAT3
      99.85%
AS1810722    
STAT6, IC50: 1.9 nM
  98.10%
Peramivir
STAT3
      99.94%
Fezakinumab
STAT3
      99.9%
BD750  
STAT5
    99.02%
Atractylenolide II
p-STAT3
      99.89%
STAT4-IN-1
STAT3, Ki: 5.0 μM
STAT5a, Ki: 22 μM
STAT5b, Ki: 26 μM
STAT6, Ki: 29 μM
STAT1, Ki: 3.8 μM
99.17%
Brevilin A
STAT3, IC50: 10.6 μM
      99.86%
STAT1/3-IN-1
STAT3
   
STAT1
Corynoline
p-STAT3
      98.84%
Sarilumab
p-STAT3
      99.36%
STAT3-IN-3
STAT3
      98.40%
15-keto-Prostaglandin E2
STAT3
      ≥99.0%
Flubendazole
STAT3
      99.05%
Stafia-1  
STAT5a, Ki: 10.9 μM
STAT5a, IC50: 22.2 μM
    99.39%
AK-068  
STAT5a, Ki: >1 μM
STAT5b, Ki: >500 μM
STAT6, Ki: 6 nM
  99.57%
LLL12
p-STAT3
      99.45%
CAY10594
p-STAT3
      98.64%
STAT3-IN-25
STAT3
      99.36%
HJC0152
STAT3
      99.75%
HO-3867
STAT3
      99.67%
STX-0119
STAT3, IC50: 74 μM (STAT3 transcription)
      98.40%
Serplulimab
p-STAT3
      99.30%
JMS-053
STAT3
      98.0%
Radotinib
STAT3
      99.19%
Anti-Mouse CD276/B7-H3 Antibody (MJ18)
p-STAT3
     
Garcinone C
Stat-3
      99.51%
STAT5-IN-2  
STAT5, EC50: 9 μM (in K562 cells)
STAT5, EC50: 5 μM (in KU812 cells )
    98.90%
Olokizumab
Stat-3
      99.54%
Sm4      
STAT1
99.01%
Mogrol
STAT3
      99.76%
Ginkgolic acid C17:1
STAT3
      99.80%
Telocinobufagin
STAT3
      99.93%
OSM-SMI-10B
p-STAT3
      99.70%
IST5-002  
STAT5a, IC50: 1.5 μM
STAT5b, IC50: 3.5 μM
    99.83%
Stafib-1  
STAT5b, IC50: 154 nM
    99.25%
Broussonin E
STAT3
      98.11%
Phellodendrine chloride
STAT3
      99.68%
NSC-370284
STAT3
STAT5
    99.27%
Cenisertib  
STAT5
    99.86%
GMB-475  
STAT5
    98.69%
Garcinone D
p-STAT3
      99.30%
Protosappanin A
STAT3
      99.95%
inS3-54A18
STAT3
      99.93%
Perindopril erbumine
STAT3
      99.98%
Medrysone    
STAT6
  99.79%
SB02024      
STAT1
99.70%
LL-K8-22      
STAT1
99.06%
Corylifol A
STAT3, IC50: 0.81 μM
      99.90%
Tetramethylcurcumin
STAT3
      99.91%
Anthraquinone-2-carboxylic acid      
STAT1
98.0%
AS2863619 free base  
STAT5
    99.87%
SD-436
STAT3, IC50: 19 nM
STAT5, IC50: >10 μM
STAT6, IC50: >10 μM
STAT1, IC50: 270 nM
98.27%
Picroside I    
STAT6
  99.48%
STAT3-IN-12
STAT3
      99.87%
YMU1
STAT3
      99.19%
Equisetin
STAT3
      99.40%
UNC1062    
STAT6
  98.92%
Ac-GpYLPQTV-NH2 acetate
STAT3, IC50: 0.33 μM
      99.00%
Reticuline
STAT3
      98.89%
PROTAC STAT6 degrader-1    
STAT6, DC50: <1 nM
  98.03%
Anti-Mouse CD106/VCAM-1 Antibody (M/K-2.7)
p-STAT3
     
Desmethoxyyangonin
STAT3
      99.00%
Graveoline
p-STAT3
      99.93%
Eflepedocokin alfa
STAT3
      ≥99.0%
WB436B
STAT3
      99.93%
Cyanidin 3,5-diglucoside chloride
STAT3
      99.44%
Triacetylresveratrol
STAT3
      99.11%
Balsalazide
STAT3
      98.65%
Fulipiftide
STAT3
      99.38%
HODHBt  
STAT5
    99.93%
HJC0416 hydrochloride
STAT3
      98.68%
Ochromycinone
STAT3
      99.61%
Golotimod hydrochloride
STAT3
      99.79%
STAT6 degrader-3    
STAT6, DC50: <1 nM
  99.26%
GSK2618960  
STAT5
   
KMR-206      
STAT1
98.86%
PROTAC FLT-3 degrader 1  
STAT5
    99.19%
Pheophytin a      
STAT1
Zharp1-211      
STAT1
99.15%
Vanicoside B
STAT3
      99.82%
ASP3026
STAT3
      99.88%
Ibrutinib-MPEA  
STAT5
    99.71%
QL-1200186
STAT3
STAT5
 
STAT1
99.95%
STAT3-IN-15
STAT3
      98.99%
Ritlecitinib tosylate
STAT3
STAT5
STAT6
  99.65%
Mulberrofuran G
STAT3
     
SZ0232
STAT3
      98.89%
OK2
p-STAT3
      99.13%
SC99
STAT3
      98.90%
Cucurbitacin IIa
STAT3
      99.90%
STAT3-IN-48
p-STAT3
      98.64%
RBN012811      
STAT1
98.79%
Balsalazide sodium hydrate
STAT3
      99.61%
STAT3-IN-17
STAT3
      98.0%
Patiromer
STAT3
STAT5
STAT6
 
CT1113  
STAT5
    99.61%
STAT6 ligand-1    
STAT6
  98.94%
Iminostilbene
STAT3
      99.34%
Polygalaxanthone III
STAT3
      99.28%
Phlorizin dihydrate
STAT3
      99.51%
MNK8
STAT3
      99.76%
ER-464195-01
STAT3
      99.72%
WB518
STAT3
p-STAT3
     
APTSTAT3-9R
STAT3
      98.82%
1-Stearoyl-sn-glycero-3-phosphocholine-d35
p-STAT3
      99%
Bellidifolin
STAT3
      99.74%
ENMD-1198
STAT3
      98.87%
UC-514321
STAT3
STAT5
    98.0%
PROTAC JAK1/2 degrader-1
STAT3
      99.47%
SH5-07
STAT3, IC50: 3.9 μM
      98.0%
Phellodendrine
STAT3
      99.60%
BP79
STAT3
 
STAT6
 
SD-1029
STAT3
     
Galiellalactone
STAT3, IC50: 250-500 nM
      99%
Cyclanoline chloride
STAT3
     
Momordicine I
STAT3
     
15(R)-Lipoxin A4
STAT3
 
STAT6
  98.3%
Globulol
STAT3
      99.74%
ZDZ-553      
STAT1, IC50: 0.87 μM
Mocravimod
STAT3
      98.39%
DCZ3301
p-STAT3
      99.73%
STAT3-IN-37
STAT3
     
Pimozide-d4
STAT3
STAT5
    99.2%
Isocryptotanshinone
STAT3
      ≥98.0%
PROTAC SKP2 Degrader-1      
STAT1
INCA033989
STAT3
STAT5
   
Guanosine 5'-diphosphate
Stat-3
     
HJC0123
STAT3
      99.06%
SD-2301
STAT3
     
Golotimod
STAT3
      98.04%
S3I-1757
Stat-3
      99.51%
ROCK2-IN-12
p-STAT3
      98.02%
STAT3-D11-PROTAC-VHL
STAT3
     
STAT3-IN-52
STAT3, Ki: 440 nM
     
SD-91
STAT3, Ki: 5.5 nM
STAT3, Kd: 28 nM
     
Ac-GpYLPQTV-NH2
STAT3, IC50: 0.33 μM
      99.38%
Biflorin      
STAT1
99.54%
Stafia-1-dipivaloyloxymethyl ester  
STAT5a
   
Eupalinolide K
STAT3
      99.20%
IMC-EB10  
STAT5
   
XOMA-213  
STAT5
    98.46%
Leucrose    
STAT6
  98.53%
Niclosamide monohydrate
STAT3, IC50: 0.25 μM (in HeLa cells)
     
SD-1008
STAT3
      99.10%
KT-333 ammonium
STAT3
      99.48%
Ritlecitinib malonate
STAT3
STAT5
STAT6
 
YYSW001
STAT3
 
STAT6
 
STAT6 degrader-4    
STAT6, DC50: < 1 nM
 
STAT3-IN-8
STAT3
     
KT-333 diammonium
STAT3
     
YSY01A
Stat-3
     
WYE-151650  
STAT5
   
c-Met-IN-24
STAT3, IC50: 4.7 μM
     
(14S,15R)-14-Deoxyoxacyclododecindione    
STAT6, IC50: 20 nM
 
DM245
p-STAT3
     
STAT3 HiBiT degrader 1
STAT3
     
STAT3-IN-38
STAT3, Kd: 45.33 μM
     
STAT3-IN-29
STAT3
     
VEGFR-2/STAT-3-IN-1
STAT3, IC50: 5.63 nM
     
STAT3-IN-49
STAT3
     
Avicin D
p-STAT3
     
P-gp-IN-36
STAT3
     
8α-Tigloyloxyhirsutinolide 13-O-acetate
STAT3
     
CPA-7
Stat-3
     
KB-0118
STAT3
     
G721-0282
p-STAT3
      99.96%
WR-S-462
STAT3, Kd: 58 nM
     
EC-70124
STAT3
     
JAK1/STAT3-IN-1
STAT3
     
FLT3-IN-28  
STAT5
   
CDK8-IN-2      
STAT1
CHI3L1-IN-4
p-STAT3
     
BRD4-IN-41
STAT3
     
MEAP
STAT3
     
JAK1-IN-20
STAT3
     
YN11
STAT3, Ki: 11.9 μM
     
WP1193
STAT3
     
Crispene E
STAT3
     
DM243
p-STAT3
     
STAT6-IN-7    
STAT6
  99.53%
STAT3/AKT-IN-1
Stat-3
     
Fa-Au      
STAT1
ROCK2-IN-7
Stat-3
     
PHI-501
STAT3
     
EGFR kinase-IN-8
STAT3
     
Anti-inflammatory agent 92
STAT3
     
ODZ10117
STAT3, IC50: 7.5 μM
     
STAT3-IN-41
STAT3
     
(trans)-STAT6-IN-13
Stat-3, IC50: 30-3000 nM
 
STAT6, IC50: ≤300 nM
 
Golotimod TFA
STAT3
     
BAY-356      
STAT1
JAK2-IN-18  
STAT5
   
HJC0416
STAT3
     
TU-100
STAT3
     
JAK2-IN-13
STAT3
STAT5
   
mTOR-IN-29
STAT3
     
STAT3-IN-46
STAT3, Kd: 323.3 nM
     
PROTAC JAK2 degrader-1
p-STAT3
STAT5
   
HAT-SIL-TG-1&AT
STAT3
STAT5
   
MLS-2384 free base
STAT3
     
ITA-5      
STAT1
STAT3/NF-κB-IN-1
STAT3, IC50: 5.86 μM
     
FLT3-IN-41  
STAT5
   
Apoptosis inducer 55
STAT3
   
STAT1
STAT3-IN-47
STAT3
     
SD-965
STAT3, DC50: 0.14 μM
     
STAT6-IN-8    
STAT6
 
7-epi-Isogarcinol
STAT3
     
STAT6 degrader-1    
STAT6
 
Orazipone      
STAT1
Lss-11
STAT3
     
STAT6-IN-9    
STAT6, EC50: 4 nM
  98.11%
PROTAC STAT6 degrader-2    
STAT6
 
STAT3-IN-44
STAT3
     
Cernuumolide J
Stat-3
     
Atractylenolide II (Standard)
p-STAT3
     
PROTAC ALK degrader-5
STAT3
     
Antitumor agent-73
STAT3
     
Glucocorticoid receptor/IL-6-IN-1
STAT3
     
N-Deacetyl-SI-109-(OEt)2
STAT3
     
NSC-368262
STAT3
     
STAT3-IN-5
p-STAT3, EC50: 170 nM
     
K882
Stat-3
     
SC-60
STAT3
     
STAT3-IN-32
STAT3
     
PTPN2/1-IN-4      
STAT1
STAT6-IN-12    
STAT6, IC50: 50 nM
 
NVP-BVB808  
STAT5
   
Hsp110-STAT3 PPI-IN-2
STAT3
     
STAT3-IN-43
STAT3, IC50: 40.7 μM
     
TPST2-IN-1      
STAT1
PDGFRA/CAIX/XII-IN-1
STAT3
     
MMP-2/9-IN-2
STAT3
     
PROTAC STAT6 degrader-4    
STAT6, DC50: 0.04 nM
 
VS1150  
STAT5
   
FLT3-IN-32 hydrochloride  
STAT5
   
Z169667518
STAT3
     
STAT3/CAIX-IN-1
STAT3, Kd: 60.03 μM
     
STAT3-IN-9
STAT3
     
NTZ-24
STAT3, IC50: 0.8 μM
     
STAT3-IN-53
STAT3, Kd: 6.16 μM
     
PROTAC STAT3 degrader-2
STAT3, ID50: 3.54 μM
     
KSI-028      
STAT1
STAT3-IN-51
STAT3
     
Ascochlorin
STAT3
     
TAVO101  
STAT5
   
NSC 850745
Stat-3, IC50: 670 nM
     
Tyk2-IN-22-d3  
STAT5
   
JAK2-IN-21
STAT3
STAT5
   
PI3K/Akt/mTOR-IN-7
STAT3
     
CHI3L1-IN-7
STAT3
     
PROTAC c-Met degrader-5
p-STAT3
     
S3D5
STAT3, Kd: 4.35 μM
     
AUH-6-96
STAT3
     
JAK2/STAT3-IN-2
STAT3
     
NW16
STAT3, Kd: 11.0 μM
     
MRC-G-001
STAT3
     
STAT3-IN-33
STAT3
     
CDK6/9-IN-2
STAT3
     
PKM2 activator 11
STAT3
     
pro-FTY
p-STAT3
     
JAK2-IN-14  
STAT5
   
Cyanidin 3,5-diglucoside chloride (Standard)
STAT3
     
XL-20      
STAT1
Furowanin A
STAT3
     
STAT6-IN-13
STAT3, IC50: 3-30 μM
 
STAT6, IC50: ≤300 nM
 
(Rac)-8-Gingerol
p-STAT3
     
CHI3L1-IN-6
STAT3
     
FLC-8  
STAT5
   
Bufothionine
p-STAT3
     
Antitumor agent-195
STAT3, IC50: 0.52 μM
     
ALOX5 stabilizer-1
STAT3
     
Geranylgeranyl pyrophosphate  
STAT5
   
STAT-3/c-Src-IN-1
STAT3, IC50: 0.844 μM
     
ITA-9      
STAT1
STAT3-IN-10
STAT3, IC50: 5.18 μM
     
Balsalazide disodium
STAT3
     
Cyclo(L-Ile-D-Leu)
STAT3
     
GYY4137 (GMP)
Stat-3
     
CHMFL-48  
STAT5
   
DETD-35
Stat-3
     
Isocucurbitacin B
STAT3
      98.98%
STAT3-IN-39
STAT3
     
Pulchinenoside E2
STAT3
      99.28%
Madindoline A
Stat-3
     
Betavulgarin
p-STAT3
     
Plumericin
STAT3
     
TM-233
Stat-3
     
ENT-03
STAT3
     
BP-1-108  
STAT5, Ki: 8.3 μM
   
PMMB-187
Stat-3, IC50: 1.81 μM