1. Signaling Pathways
  2. Protein Tyrosine Kinase/RTK
  3. TAM Receptor
  4. TAM Receptor Inhibitors

TAM Receptor Inhibitors

Axl

Mer

Tyro3

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

TAM Receptor Inhibitors
Product Name Axl Mer Tyro3 Purity
Bemcentinib
Axl
    99.92%
Cabozantinib
Axl
    99.97%
Gilteritinib
Axl
    99.84%
2-D08
Axl
    99.37%
BMS 777607
Axl
 
Tyro3
99.36%
Ladarutatug
Axl
   
TAM-IN-1
Axl, Ki: 130 pM
Mer, Ki: <50 pM
 
UNC2250
Axl
Mer
  99.92%
Zanzalintinib
Axl
Mer
  99.91%
LDC1267
Axl, IC50: 42 nM
MERTK, IC50: 130 nM
Tyro3, IC50: 63 nM
99.64%
Dubermatinib
Axl
    99.84%
UNC569
Axl
Mer
Tyro3
99.92%
UNC5293
Axl
 
Tyro3
99.93%
Gilteritinib hemifumarate
Axl
    99.75%
UNC2541  
Mer
  99.71%
Tamnorzatinib
Axl
Mer
Tyro3
98.59%
Batiraxcept
Axl
    99.91%
CEP-40783
Axl
    99.61%
SGI-7079
Axl
    99.32%
Tilvestamab
Axl
    98.08%
UNC1062
Axl, : 85 nM
 
Tyro3, : 60 nM
98.92%
NPS-1034
Axl
    98.0%
UNC9426
Axl, IC50: 190 nM
MERTK, IC50: 580 nM
Tyro3, IC50: 2.1 nM
99.51%
RU-302
Axl
    98.72%
UNC2881
Axl
Mer
  99.79%
Enapotamab
Axl
    99.9%
Ningetinib
Axl
    99.82%
Mecbotamab
Axl
    99.83%
PF-07265807
Axl, IC50: 0.9 nM
Mer, IC50: 2.3 nM
Tyro3, IC50: 6 nM
Adrixetinib
Axl, Kd: 0.3 nM
Mer, Kd: 0.8 nM
  99.55%
UNC4203
Axl
 
Tyro3
99.80%
AZ14145845
Axl
Mer
  98.00%
DS-1205b free base
Axl
Mer
  99.92%
PROTAC Axl Degrader 2
Axl
    98.01%
Cabozantinib-d6
Axl
    98.14%
AXL-IN-13
Axl
    98.03%
Ningetinib Tosylate
Axl
    99.59%
Adrixetinib TFA
Axl, Kd: 0.3 nM
Mer, Kd: 0.8 nM
  99.82%
Mipasetamab
Axl
    98.26%
TL4830031
Axl
    ≥98.0%
AG01
Axl
   
Cabozantinib hydrochloride
Axl
   
Axl-IN-6
Axl
   
UNC8212
Axl, IC50: 1.3 nM
MERTK, IC50: 1.5 nM
Tyro3, IC50: 6.7 nM
Axl-IN-9
Axl
   
Axl-IN-11
Axl
   
PROTAC Axl Degrader 1
Axl
   
Axl-IN-4
Axl
   
Axl-IN-17
Axl, IC50: 3.23 nM
Mer
Tyro3
Axl-IN-10
Axl
   
Bemcentinib (GMP)
Axl
   
HIV-IN-7
Axl
   
Axl/Mer/CSF1R-IN-1
Axl
Mer
 
Axl-IN-21
Axl, IC50: 4 nM
Axl, Kd: 2.7 nM
Mer, Kd: 1.4 nM
 
UNC3133
Axl, IC50: 17 nM
MERTK, IC50: 3.0 nM
Tyro3, IC50: 31 nM
Axl-IN-12
Axl
   
AXL-IN-15
Axl
   
Axl-IN-7
Axl
   
NTQ2494
Axl, IC50: 4.89 nM
   
Axl-IN-19
Axl, IC50: 5.3 nM
   
Axl-IN-16
Axl
   
Axl-IN-8
Axl
   
Anticancer agent 109
Axl
   
Axl-IN-3
Axl
   
R916562
Axl
   
AXL-IN-14
Axl
   
Axl-IN-5
Axl