MDA7
MDA7 is the selective agonist for cannabinoid receptor 2 with EC50 of 128 nM and 67.4 nM in human CB2 receptor and rat CB2 receptor. MDA7 exhibits good affinity to human CB2 receptor and rat CB2 receptor with Ki of 422 nM and 238 nM. MDA7 exhibits analgesic activity in rats models.
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- CAS. Nr.: 1103840-28-3
- Formel: C22H25NO2
- Molecular Weight:335.44
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Speicherung:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biologische Aktivität
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rat CB2-R 67.4 nM (IC50) |
hCB2-R 128 nM (IC50) |
rat CB2-R 238 nM (Ki) |
hCB2-R 422 nM (Ki) |
rCB1-R 2565 nM (Ki) |
Chemical Information
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CAS. Nr. 1103840-28-3
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Molecular Weight 335.44
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Formel C22H25NO2
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SMILES
O=C(N1CCCCC1)C2=CC=C3C(OCC3(CC4=CC=CC=C4)C)=C2
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Versand
Room temperature in continental US; may vary elsewhere.
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Speicherung
Please store the product under the recommended conditions in the Certificate of Analysis.
Reinheit & Dokumentation
Verweise
Calculators
Konzentration (Stammlösung) × Volumen (Stammlösung) = Konzentration (Ziellösung) × Volumen (Ziellösung)