CDK9-IN-52
CDK9-IN-52 is a CDK9 inhibitor. CDK9-IN-52 exhibits antiproliferative activity against cancer cells. CDK9-IN-52 can be used in studies related to lung cancer, cervical cancer, and breast cancer.
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- Formule: C24H17F2N3O
- Masse moléculaire:401.41
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Activité biologique
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Chemical Information
- Pureté et documentation
- Références
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Help & FAQs
Activité biologique
Description
IC50 & Target
[1]|
CDK9 |
In Vitro
CDK9-IN-52 (D6) potently inhibits the proliferation of HeLa, A549, SiHa and MCF-7 cancer cells with IC50 values of 6.64, 7.27, 10.36 and 10.82 μM, respectively. Meanwhile, it exhibits selective cytotoxicity toward cancer cells compared with normal HEK-293t cells, with the highest selectivity against HeLa cells (SI=9.1)[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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Masse moléculaire 401.41
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Formule C24H17F2N3O
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SMILES
N#CC1=CC(C(C=C2)=CC(F)=C2NC(CCN3C(C=CC(F)=C4)=C4C=C3)=O)=CC=C1
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
CDK9-IN-52 Related Classifications
HY-183699 Related Classifications
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