104860-61-9
Chemical Structure
R 50595 hydrochloride
- CAS No.: 104860-61-9
- Formula:C30H35Cl2F2N3O3
- Molecular Weight:594.52
IUPAC Name: 4-amino-N-((3S,4S)-1-(4,4-bis(4-fluorophenyl)butyl)-3-methoxypiperidin-4-yl)-5-chloro-2-methoxybenzamide hydrochloride
InChIKey: ODGIHIUVACVQTA-YDFTWFOHSA-N
SMILES: O=C(N[C@@H]1[C@@H](OC)CN(CCCC(C2=CC=C(F)C=C2)C3=CC=C(F)C=C3)CC1)C4=CC(Cl)=C(N)C=C4OC.[H]Cl
Biological Activity: 50595 hydrochloride is a selective noncompetitive cisapride antagonist that interferes with the activity of cisapride and BRL 24924. R 50595 hydrochloride has no effect on the response to electrical stimulation at concentrations up to 3 X 10(-7) M. R 50595 hydrochloride antagonizes the effects of cisapride and BRL 24924 in a noncompetitive manner. R 50595 hydrochloride completely abolishes the effects of 5-HT at a concentration of 3 X 10(-7) M and also antagonizes the effects of 5-HT in a noncompetitive manner[1].
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R 50595 hydrochloride | 50595 hydrochloride is a selective noncompetitive cisapride antagonist that interferes with the activity of cisapride and BRL 24924. R 50595 hydrochloride has no effect on the response to electrical stimulation at concentrations up to 3 X 10(-7) M. R 50595 hydrochloride antagonizes the effects of cisapride and BRL 24924 in a noncompetitive manner. R 50595 hydrochloride completely abolishes the effects of 5-HT at a concentration of 3 X 10(-7) M and also antagonizes the effects of 5-HT in a noncompetitive manner. | |||||||||||||||||||||
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