1110883-26-5
Chemical Structure
ID110460001
- CAS No.: 1110883-26-5
- Formula:C20H24N2O3
- Molecular Weight:340.42
IUPAC Name: 2-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-N-(2-(dimethylamino)-2-phenylethyl)acetamide
InChIKey: LWZACHFUFUKWNQ-UHFFFAOYSA-N
SMILES: O=C(NCC(C=1C=CC=CC1)N(C)C)CC2=CC=C3OCCOC3=C2
Biological Activity: ID110460001 is a full agonist of μ-opioid receptor and an agonist of δ-opioid receptor. ID110460001 exhibits high intrinsic efficacy for G protein pathway activation of μ-opioid receptor, and this property is not affected by the reduction in receptor quantity. ID110460001 acts only as a very weak partial agonist in the β-arrestin-2 pathway of both receptors, and binds to μ-opioid receptor via a specific mode. The efficacy of ID110460001 in the G protein pathway of δ-opioid receptor is sensitive to changes in receptor quantity. ID110460001 can be used in pain-related research[1].
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ID110460001 | ID110460001 is a full agonist of μ-opioid receptor and an agonist of δ-opioid receptor. ID110460001 exhibits high intrinsic efficacy for G protein pathway activation of μ-opioid receptor, and this property is not affected by the reduction in receptor quantity. ID110460001 acts only as a very weak partial agonist in the β-arrestin-2 pathway of both receptors, and binds to μ-opioid receptor via a specific mode. The efficacy of ID110460001 in the G protein pathway of δ-opioid receptor is sensitive to changes in receptor quantity. ID110460001 can be used in pain-related research. | |||||||||||||||||||||
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Keywords
