1132641-75-8
1132641-75-8
Chemical Structure
Telcagepant-d8
Synonym(s): MK-0974-d8
- CAS No.: 1132641-75-8
- Formula:C26H19D8F5N6O3
- Molecular Weight:574.57
InChIKey: CGDZXLJGHVKVIE-CSFDOCDKSA-N
SMILES: O=C1N(C2C([2H])([2H])C([2H])([2H])N(C([2H])([2H])C2([2H])[2H])C(N[C@H]3C(N(C[C@H](C4=C(C(F)=CC=C4)F)CC3)CC(F)(F)F)=O)=O)C5=CC=CN=C5N1
Biological Activity: Telcagepant-d8 (MK-0974-d8) is deuterium labeled Telcagepant. Telcagepant (MK-0974) is an orally active calcitonin gene-related peptide (CGRP) receptor antagonist with Kis of 0.77 nM and 1.2 nM for human and rhesus CGRP receptors, respectively.
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Telcagepant-d8 | Telcagepant-d8 (MK-0974-d8) is deuterium labeled Telcagepant. Telcagepant (MK-0974) is an orally active calcitonin gene-related peptide (CGRP) receptor antagonist with Kis of 0.77 nM and 1.2 nM for human and rhesus CGRP receptors, respectively. | |||||||||||||||||||||
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Telcagepant | 98.63% | Telcagepant (MK-0974) is an orally active calcitonin gene-related peptide (CGRP) receptor antagonist with Kis of 0.77 nM and 1.2 nM for human and rhesus CGRP receptors, respectively. | ||||||||||||||||||||
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Keywords
