1133705-99-3
1133705-99-3
Chemical Structure
GSK172981
- CAS No.: 1133705-99-3
- Formula:C26H22FN3O
- Molecular Weight:411.47
IUPAC Name: (S)-3-amino-N-(cyclopropyl(phenyl)methyl)-2-(3-fluorophenyl)quinoline-4-carboxamide
InChIKey: ZKGNLARKIMWKFE-XMMPIXPASA-N
SMILES: O=C(N[C@H](C1=CC=CC=C1)C2CC2)C3=C(C(C4=CC=CC(F)=C4)=NC5=CC=CC=C35)N
Biological Activity: GSK172981 is a brain-penetrant tachykinin NK3 receptor antagonist with pKi values of 7.7 and 7.8 for human and native guinea pig NK3 receptors, respectively. GSK172981 can be used for the study of schizophrenia[1].
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GSK172981 | GSK172981 is a brain-penetrant tachykinin NK3 receptor antagonist with pKi values of 7.7 and 7.8 for human and native guinea pig NK3 receptors, respectively. GSK172981 can be used for the study of schizophrenia. | |||||||||||||||||||||
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References
Keywords
