1189574-93-3
1189574-93-3
Chemical Structure
Loperamide-d6
Synonym(s): ADL 2-1294-d6
- CAS No.: 1189574-93-3
- Formula:C29H27D6ClN2O2
- Molecular Weight:483.07
IUPAC Name: 3,5-diiodo-4-methylpyridin-2-amine
InChIKey: RDOIQAHITMMDAJ-WFGJKAKNSA-N
SMILES: OC(CC1)(C2=CC=C(C=C2)Cl)CCN1CCC(C3=CC=CC=C3)(C4=CC=CC=C4)C(N(C([2H])([2H])[2H])C([2H])([2H])[2H])=O
Biological Activity: Loperamide-d6 is the deuterium labeled Loperamide[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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Loperamide-d6 | 98.88% | Loperamide-d6 is the deuterium labeled Loperamide. | ||||||||||||||||||||
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Loperamide | 99.85% | Loperamide (ADL 2-1294) is selective and orally active μ opioid receptor agonist with Ki valuess of 3, 48 and 1156 nM against μ, δ and κ opioid receptor, respectively. Loperamide produces antinociception and antihyperalgesia. Loperamide exhibits peripheral selectivity, enhancing fluid, electrolyte, and glucose absorption, reversing PGE2 (HY-101952)- and Cholera toxin (HY-P1446)-induced intestinal secretion, and reducing intestinal motility. Loperamide can be used for the researches of inflammatory pain and protracted diarrhoea. | ||||||||||||||||||||
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References
Keywords
