138562-23-9
Chemical Structure
RP-69758
- CAS No.: 138562-23-9
- Formula:C26H26N4O5
- Molecular Weight:474.51
IUPAC Name: 2-(3-(3-(2-((2-(methyl(phenyl)amino)-2-oxoethyl)(phenyl)amino)-2-oxoethyl)ureido)phenyl)acetic acid
InChIKey: CRUWRCOXWORZBA-UHFFFAOYSA-N
SMILES: O=C(CC1=CC=CC(NC(NCC(N(C2=CC=CC=C2)CC(N(C3=CC=CC=C3)C)=O)=O)=O)=C1)O
Biological Activity: RP-69758 is a potent and selective non-peptide cholecystokinin-B (CCKB)/gastrin receptor antagonist. RP-69758 exhibits >200-fold selectivity for CCKB over CCKA receptors. RP-69758 antagonizes CCK-8-induced neuronal firing in rat hippocampal slices. RP-69758 inhibits Pentagastrin (HY-A0261)-induced gastric acid secretion in the rat. RP-69758 can be used for neurological disorders and gastrointestinal disease research[1].
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RP-69758 | RP-69758 is a potent and selective non-peptide cholecystokinin-B (CCKB)/gastrin receptor antagonist. RP-69758 exhibits >200-fold selectivity for CCKB over CCKA receptors. RP-69758 antagonizes CCK-8-induced neuronal firing in rat hippocampal slices. RP-69758 inhibits Pentagastrin (HY-A0261)-induced gastric acid secretion in the rat. RP-69758 can be used for neurological disorders and gastrointestinal disease research. | |||||||||||||||||||||
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Keywords
