1403258-69-4
1403258-69-4
Chemical Structure
EZH2-IN-5
- CAS No.: 1403258-69-4
- Formula:C26H37BrN4O2
- Molecular Weight:517.50
IUPAC Name: 5-bromo-N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-3-(((1r,4r)-4-(dimethylamino)cyclohexyl)(ethyl)amino)-2-methylbenzamide
InChIKey: FKKHGOZTTQASQA-MEMLXQNLSA-N
SMILES: CCN([C@H]1CC[C@@H](CC1)N(C)C)C2=C(C(C(NCC3=C(C=C(NC3=O)C)C)=O)=CC(Br)=C2)C
Biological Activity: EZH2-IN-5 is a potent EZH2 inhibitor with IC50 values of 1.52 nM and 4.07 nM for wild-type and mutant Tyr641 EZH2, respectively[1].
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EZH2-IN-5 | EZH2-IN-5 is a potent EZH2 inhibitor with IC50 values of 1.52 nM and 4.07 nM for wild-type and mutant Tyr641 EZH2, respectively. | |||||||||||||||||||||
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References
Keywords
