140924-11-4
140924-11-4
Chemical Structure
AP-238
- CAS No.: 140924-11-4
- Formula:C18H26N2O
- Molecular Weight:286.41
InChIKey: JELNWDOXWGBBLO-QJBCGIKSSA-N
SMILES: CCC(N1[C@H](C)CN(C/C=C/C2=CC=CC=C2)C[C@@H]1C)=O
Biological Activity: AP-238 is a a new synthetic opioid (NSO), and acts as an agonist for μ-opioid receptor (MOR) with an EC50 of 248 nM. AP-238 exhibits analgesic activity[1][2].
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AP-238 | AP-238 is a a new synthetic opioid (NSO), and acts as an agonist for μ-opioid receptor (MOR) with an EC50 of 248 nM. AP-238 exhibits analgesic activity. | |||||||||||||||||||||
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References
- [1]. Jurowski K, et, al. Prediction of key toxicity endpoints of AP-238 a new psychoactive substance for clinical toxicology and forensic purposes using in silico methods. Sci Rep. 2024 Nov 22;14(1):28977. [Content Brief]
- [2]. Brunetti P, et al., Human metabolism and basic pharmacokinetic evaluation of AP-238: A recently emerged acylpiperazine opioid. Drug Test Anal. 2024 Feb;16(2):221-235. [Content Brief]
Keywords
